| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Fatty acid-binding protein, adipocyte |
|---|
| Ligand | BDBM312471 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Time Resolved-Fluorescence Energy Transfer (TR-FRET) Assay |
|---|
| IC50 | 9.00±n/a nM |
|---|
| Citation |  Buettelmann, B; Ceccarelli, SM; Kuehne, H; Kuhn, B; Neidhart, W; Obst Sander, U; Richter, H Bicyclic thiophenylamide compounds US Patent US9604977 Publication Date 3/28/2017 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Fatty acid-binding protein, adipocyte |
|---|
| Name: | Fatty acid-binding protein, adipocyte |
|---|
| Synonyms: | A-FABP | AFABP | ALBP | Adipocyte lipid-binding protein | FABP4 | FABP4_HUMAN | Fatty acid binding protein adipocyte | Fatty acid-binding protein 4 | Fatty acid-binding protein 4 (FABP4) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 14719.23 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P15090 |
|---|
| Residue: | 132 |
|---|
| Sequence: | MCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKN
TEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVM
KGVTSTRVYERA
|
|
|
|---|
| BDBM312471 |
|---|
| n/a |
|---|
| Name | BDBM312471 |
|---|
| Synonyms: | 2-[5-(3-Cyclopropyl-[1,2,4]oxadiazol-5-yl)-3,4-dihydro-2H-thieno[2,3-b]pyran-6-ylcarbamoyl]-cyclopent-1-enecarboxylic acid | US9604977, Example 217 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H19N3O5S |
|---|
| Mol. Mass. | 401.436 |
|---|
| SMILES | OC(=O)C1=C(CCC1)C(=O)Nc1sc2OCCCc2c1-c1nc(no1)C1CC1 |t:3| |
|---|
| Structure | 
|
|---|
Search and Browse
