Reaction Details |
| Report a problem with these data |
Target | Casein kinase I isoform alpha |
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Ligand | BDBM10842 |
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Substrate/Competitor | Casein |
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Meas. Tech. | Kinase Inhibition Assay |
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Temperature | 303.15±n/a K |
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IC50 | 400±n/a nM |
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Comments | extracted |
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Citation | Gompel, M; Leost, M; De Kier Joffe, EB; Puricelli, L; Franco, LH; Palermo, J; Meijer, L Meridianins, a new family of protein kinase inhibitors isolated from the ascidian Aplidium meridianum. Bioorg Med Chem Lett14:1703-7 (2004) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Casein kinase I isoform alpha |
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Name: | Casein kinase I isoform alpha |
Synonyms: | CK1 | CKI-alpha | Casein Kinase I | Csnk1a1 | KC1A_RAT |
Type: | Enzyme |
Mol. Mass.: | 37514.97 |
Organism: | Rattus norvegicus (rat) |
Description: | n/a |
Residue: | 325 |
Sequence: | MASSSGSKAEFIVGGKYKLVRKIGSGSFGDIYLAINITNGEEVAVKLESQKARHPQLLYE
SKLYKILQGGVGIPHIRWYGQGKDYNVLVMDLLGPSLEDLFNFCSRRFTMKTVLMLADQM
ISRIEYVHTKNFIHRDIKPDNFLMGIGRHCNKLFLIDFGLAKKYRDNRTRQHIPYREDKN
LTGTARYASINAHLGIEQSRRDDMESLGYVLMYFNRTSLPWQGLKAATKKQKYEKISEKK
MSTPVEVLCKGFPAEFAMYLNYCRGLRFEEAPDYMYLRQLFRILFRTLNHQYDYTFDWTM
LKQKAAQQAASSSGQGQQAQTPTGF
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BDBM10842 |
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Casein |
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Name: | Casein |
Synonyms: | n/a |
Type: | Other Protein Type |
Mol. Mass.: | 20807.68 |
Organism: | Homo sapiens (Human) |
Description: | n/a |
Residue: | 177 |
Sequence: | MRLLILTCLVAVALARPKLPLRYPERLQNPSESSEPIPLESREEYMNGMNRQRNILREKQ
TDEIKDTRNESTQNCVVAESEKMESSISSSSEEQFCRLNEYNQLQLQAAHAQEQIRRMNE
NSHVQVPFQQLNQLAAYPYAVWYYPQIMQYVPFPPFSDISNPTAHENYEKNNVMLQW
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