Reaction Details |
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Target | Casein kinase II subunit alpha |
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Ligand | BDBM11318 |
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Substrate/Competitor | CK-2 Peptide Substrate |
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Meas. Tech. | Kinase Inhibition Assay |
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pH | 7.5±n/a |
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Temperature | 295.15±n/a K |
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Ki | 1850±n/a nM |
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Citation | De Moliner, E; Moro, S; Sarno, S; Zagotto, G; Zanotti, G; Pinna, LA; Battistutta, R Inhibition of protein kinase CK2 by anthraquinone-related compounds. A structural insight. J Biol Chem278:1831-6 (2003) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Casein kinase II subunit alpha |
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Name: | Casein kinase II subunit alpha |
Synonyms: | ACK2 | CK II | CK2- alpha | CSK2A_MAIZE | Casein Kinase II |
Type: | Enzyme |
Mol. Mass.: | 39238.74 |
Organism: | Zea mays (Maize) |
Description: | n/a |
Residue: | 332 |
Sequence: | MSKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKC
IIKILKPVKKKKIKREIKILQNLCGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLY
PTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPG
KEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKI
AKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLL
RYDHQERLTALEAMTHPYFQQVRAAENSRTRA
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BDBM11318 |
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CK-2 Peptide Substrate |
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Name: | CK-2 Peptide Substrate |
Synonyms: | n/a |
Type: | Peptide |
Mol. Mass.: | 1446.31 |
Organism: | n/a |
Description: | n/a |
Residue: | 12 |
Sequence: | |