| Reaction Details |
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 | Report a problem with these data |
| Target | Sentrin-specific protease 7 |
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| Ligand | BDBM103829 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Binding Assay |
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| IC50 | 3400±1500 nM |
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| Citation |  Chen, Y Methods of identifying SENP1 inhibitors US Patent US9791447 Publication Date 10/17/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| Sentrin-specific protease 7 |
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| Name: | Sentrin-specific protease 7 |
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| Synonyms: | KIAA1707 | SENP7 | SENP7_HUMAN | SSP2 | SUSP2 | Sentrin-specific protease 7 (SENP7) |
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| Type: | Protein |
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| Mol. Mass.: | 119657.39 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q9BQF6 |
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| Residue: | 1050 |
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| Sequence: | MDKRKLGRRPSSSEIITEGKRKKSSSDLSEIRKMLNAKPEDVHVQSPLSKFRSSERWTLP
LQWERSLRNKVISLDHKNKKHIRGCPVTSKSSPERQLKVMLTNVLWTDLGRKFRKTLPRN
DANLCDANKVQSDSLPSTSVDSLETCQKLEPLRQSLNLSERIPRVILTNVLGTELGRKYI
RTPPVTEGSLSDTDNLQSEQLSSSSDGSLESYQNLNPHKSCYLSERGSQRSKTVDDNSAK
QTAHNKEKRRKDDGISLLISDTQPEDLNSGSRGCDHLEQESRNKDVKYSDSKVELTLISR
KTKRRLRNNLPDSQYCTSLDKSTEQTKKQEDDSTISTEFEKPSENYHQDPKLPEEITTKP
TKSDFTKLSSLNSQELTLSNATKSASAGSTTETVENSNSIDIVGISSLVEKDENELNTIE
KPILRGHNEGNQSLISAEPIVVSSDEEGPVEHKSSEILKLQSKQDRETTNENESTSESAL
LELPLITCESVQMSSELCPYNPVMENISSIMPSNEMDLQLDFIFTSVYIGKIKGASKGCV
TITKKYIKIPFQVSLNEISLLVDTTHLKRFGLWKSKDDNHSKRSHAILFFWVSSDYLQEI
QTQLEHSVLSQQSKSSEFIFLELHNPVSQREELKLKDIMTEISIISGELELSYPLSWVQA
FPLFQNLSSKESSFIHYYCVSTCSFPAGVAVAEEMKLKSVSQPSNTDAAKPTYTFLQKQS
SGCYSLSITSNPDEEWREVRHTGLVQKLIVYPPPPTKGGLGVTNEDLECLEEGEFLNDVI
IDFYLKYLILEKASDELVERSHIFSSFFYKCLTRKENNLTEDNPNLSMAQRRHKRVRTWT
RHINIFNKDYIFVPVNESSHWYLAVICFPWLEEAVYEDFPQTVSQQSQAQQSQNDNKTID
NDLRTTSTLSLSAEDSQSTESNMSVPKKMCKRPCILILDSLKAASVQNTVQNLREYLEVE
WEVKLKTHRQFSKTNMVDLCPKVPKQDNSSDCGVYLLQYVESFFKDPIVNFELPIHLEKW
FPRHVIKTKREDIRELILKLHLQQQKGSSS
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| BDBM103829 |
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| n/a |
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| Name | BDBM103829 |
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| Synonyms: | SPI-04 | US11041859, Code SPI-04 | US9791447, Compound SPI-04 |
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| Type | Small organic molecule |
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| Emp. Form. | C34H25N6O12S4 |
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| Mol. Mass. | 837.856 |
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| SMILES | Nc1ccc(\N=N\c2ccc(\C=C\c3ccc(cc3S(O)(=O)=O)\N=N\c3ccc(N)c4ccc(cc34)S([O-])(=O)=O)c(c2)S(O)(=O)=O)c2cc(ccc12)S(O)(=O)=O |
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| Structure | 
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