| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Sentrin-specific protease 7 |
|---|
| Ligand | BDBM103834 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Binding Assay |
|---|
| IC50 | 1900±2100 nM |
|---|
| Citation |  Chen, Y Methods of identifying SENP1 inhibitors US Patent US9791447 Publication Date 10/17/2017 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Sentrin-specific protease 7 |
|---|
| Name: | Sentrin-specific protease 7 |
|---|
| Synonyms: | KIAA1707 | SENP7 | SENP7_HUMAN | SSP2 | SUSP2 | Sentrin-specific protease 7 (SENP7) |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 119657.39 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | Q9BQF6 |
|---|
| Residue: | 1050 |
|---|
| Sequence: | MDKRKLGRRPSSSEIITEGKRKKSSSDLSEIRKMLNAKPEDVHVQSPLSKFRSSERWTLP
LQWERSLRNKVISLDHKNKKHIRGCPVTSKSSPERQLKVMLTNVLWTDLGRKFRKTLPRN
DANLCDANKVQSDSLPSTSVDSLETCQKLEPLRQSLNLSERIPRVILTNVLGTELGRKYI
RTPPVTEGSLSDTDNLQSEQLSSSSDGSLESYQNLNPHKSCYLSERGSQRSKTVDDNSAK
QTAHNKEKRRKDDGISLLISDTQPEDLNSGSRGCDHLEQESRNKDVKYSDSKVELTLISR
KTKRRLRNNLPDSQYCTSLDKSTEQTKKQEDDSTISTEFEKPSENYHQDPKLPEEITTKP
TKSDFTKLSSLNSQELTLSNATKSASAGSTTETVENSNSIDIVGISSLVEKDENELNTIE
KPILRGHNEGNQSLISAEPIVVSSDEEGPVEHKSSEILKLQSKQDRETTNENESTSESAL
LELPLITCESVQMSSELCPYNPVMENISSIMPSNEMDLQLDFIFTSVYIGKIKGASKGCV
TITKKYIKIPFQVSLNEISLLVDTTHLKRFGLWKSKDDNHSKRSHAILFFWVSSDYLQEI
QTQLEHSVLSQQSKSSEFIFLELHNPVSQREELKLKDIMTEISIISGELELSYPLSWVQA
FPLFQNLSSKESSFIHYYCVSTCSFPAGVAVAEEMKLKSVSQPSNTDAAKPTYTFLQKQS
SGCYSLSITSNPDEEWREVRHTGLVQKLIVYPPPPTKGGLGVTNEDLECLEEGEFLNDVI
IDFYLKYLILEKASDELVERSHIFSSFFYKCLTRKENNLTEDNPNLSMAQRRHKRVRTWT
RHINIFNKDYIFVPVNESSHWYLAVICFPWLEEAVYEDFPQTVSQQSQAQQSQNDNKTID
NDLRTTSTLSLSAEDSQSTESNMSVPKKMCKRPCILILDSLKAASVQNTVQNLREYLEVE
WEVKLKTHRQFSKTNMVDLCPKVPKQDNSSDCGVYLLQYVESFFKDPIVNFELPIHLEKW
FPRHVIKTKREDIRELILKLHLQQQKGSSS
|
|
|
|---|
| BDBM103834 |
|---|
| n/a |
|---|
| Name | BDBM103834 |
|---|
| Synonyms: | SPI-09 | US11041859, Code SPI-09 | US9791447, Compound SPI-09 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H13N3O9S3 |
|---|
| Mol. Mass. | 487.484 |
|---|
| SMILES | Nc1ccc2cc(cc(c2c1\N=N\c1ccc(cc1)S(O)(=O)=O)S(O)(=O)=O)S(O)(=O)=O |
|---|
| Structure | 
|
|---|
Search and Browse
