| Reaction Details |
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 | Report a problem with these data |
| Target | POU domain, class 2, transcription factor 2 |
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| Ligand | BDBM350836 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Inhibition Assay |
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| IC50 | 10000±n/a nM |
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| Citation |  Bacon, EM; Cai, ZR; Cottell, JJ; Ji, M; Jin, H; Lazerwith, SE; Morganelli, PA; Pyun, H Polycyclic-carbamoylpyridone compounds and their pharmaceutical use US Patent US9795602 Publication Date 10/24/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| POU domain, class 2, transcription factor 2 |
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| Name: | POU domain, class 2, transcription factor 2 |
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| Synonyms: | Lymphoid-restricted immunoglobulin octamer-binding protein NF-A2 | OCT2 | OCT2 | OTF-2 | OTF2 | Oct-2 | Octamer-binding protein 2 | Octamer-binding transcription factor 2 | Octamer-binding transcription factor 2 (OCT2) | PO2F2_HUMAN | POU domain, class 2, transcription factor 2 | POU2F2 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 51217.88 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_109671 |
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| Residue: | 479 |
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| Sequence: | MVHSSMGAPEIRMSKPLEAEKQGLDSPSEHTDTERNGPDTNHQNPQNKTSPFSVSPTGPS
TKIKAEDPSGDSAPAAPLPPQPAQPHLPQAQLMLTGSQLAGDIQQLLQLQQLVLVPGHHL
QPPAQFLLPQAQQSQPGLLPTPNLFQLPQQTQGALLTSQPRAGLPTQAVTRPTLPDPHLS
HPQPPKCLEPPSHPEEPSDLEELEQFARTFKQRRIKLGFTQGDVGLAMGKLYGNDFSQTT
ISRFEALNLSFKNMCKLKPLLEKWLNDAETMSVDSSLPSPNQLSSPSLGFDGLPGRRRKK
RTSIETNVRFALEKSFLANQKPTSEEILLIAEQLHMEKEVIRVWFCNRRQKEKRINPCSA
APMLPSPGKPASYSPHMVTPQGGAGTLPLSQASSSLSTTVTTLSSAVGTLHPSRTAGGGG
GGGGAAPPLNSIPSVTPPPPATTNSTNPSPQGSHSAIGLSGLNPSTGPGLWWNPAPYQP
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| BDBM350836 |
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| n/a |
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| Name | BDBM350836 |
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| Synonyms: | US9795602, Compound 28 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H16F3N3O4 |
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| Mol. Mass. | 407.3432 |
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| SMILES | Oc1c2C(=O)N[C@H]3CCC[C@H]3n2cc(C(=O)NCc2c(F)cc(F)cc2F)c1=O |r| |
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| Structure | 
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