| Reaction Details |
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 | Report a problem with these data |
| Target | Amine oxidase [flavin-containing] A |
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| Ligand | BDBM151625 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Monoamine Oxidase (MAO) Assay |
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| IC50 | 2100±n/a nM |
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| Citation |  Vankayalapati, H; Sorna, V; Warner, SL; Stephens, B; Bearss, DJ; Sharma, S Substituted (E)-N′-(1-phenylethylidene)benzohydrazide analogs as histone demethylase inhibitors US Patent US9555024 Publication Date 1/31/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Amine oxidase [flavin-containing] A |
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| Name: | Amine oxidase [flavin-containing] A |
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| Synonyms: | AOFA_HUMAN | Amine oxidase (flavin-containing) A | MAO-A | MAOA | Monoamine oxidase | Monoamine oxidase type A | Monoamine oxidase type A (MAO A) | Monoamine oxidase type A (MAO A) | Monoamine oxidase type A (MAOA) |
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| Type: | Protein |
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| Mol. Mass.: | 59689.53 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21397 |
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| Residue: | 527 |
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| Sequence: | MENQEKASIAGHMFDVVVIGGGISGLSAAKLLTEYGVSVLVLEARDRVGGRTYTIRNEHV
DYVDVGGAYVGPTQNRILRLSKELGIETYKVNVSERLVQYVKGKTYPFRGAFPPVWNPIA
YLDYNNLWRTIDNMGKEIPTDAPWEAQHADKWDKMTMKELIDKICWTKTARRFAYLFVNI
NVTSEPHEVSALWFLWYVKQCGGTTRIFSVTNGGQERKFVGGSGQVSERIMDLLGDQVKL
NHPVTHVDQSSDNIIIETLNHEHYECKYVINAIPPTLTAKIHFRPELPAERNQLIQRLPM
GAVIKCMMYYKEAFWKKKDYCGCMIIEDEDAPISITLDDTKPDGSLPAIMGFILARKADR
LAKLHKEIRKKKICELYAKVLGSQEALHPVHYEEKNWCEEQYSGGCYTAYFPPGIMTQYG
RVIRQPVGRIFFAGTETATKWSGYMEGAVEAGERAAREVLNGLGKVTEKDIWVQEPESKD
VPAVEITHTFWERNLPSVSGLLKIIGFSTSVTALGFVLYKYKLLPRS
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| BDBM151625 |
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| n/a |
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| Name | BDBM151625 |
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| Synonyms: | US8987335, -- |
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| Type | Small organic molecule |
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| Emp. Form. | C9H11N |
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| Mol. Mass. | 133.1903 |
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| SMILES | N[C@@H]1CC1c1ccccc1 |r| |
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| Structure | 
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