| Reaction Details |
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 | Report a problem with these data |
| Target | Free fatty acid receptor 4 |
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| Ligand | BDBM382133 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | BRET assay |
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| EC50 | 2750±n/a nM |
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| Citation |  Kumar, S; Sharma, R; Deore, VB; Yewalkar, NN Substituted phenyl alkanoic acid compounds as GPR120 agonists and uses thereof US Patent US10273230 Publication Date 4/30/2019 |
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| More Info.: | Get all data from this article, Assay Method |
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| Free fatty acid receptor 4 |
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| Name: | Free fatty acid receptor 4 |
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| Synonyms: | FFAR4 | FFAR4_HUMAN | G-protein coupled receptor 120 | G-protein coupled receptor 129 | G-protein coupled receptor GT01 | G-protein coupled receptor PGR4 | GPR120 | GPR129 | O3FAR1 | Omega-3 fatty acid receptor 1 | PGR4 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 42256.91 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1508994 |
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| Residue: | 377 |
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| Sequence: | MSPECARAAGDAPLRSLEQANRTRFPFFSDVKGDHRLVLAAVETTVLVLIFAVSLLGNVC
ALVLVARRRRRGATACLVLNLFCADLLFISAIPLVLAVRWTEAWLLGPVACHLLFYVMTL
SGSVTILTLAAVSLERMVCIVHLQRGVRGPGRRARAVLLALIWGYSAVAALPLCVFFRVV
PQRLPGADQEISICTLIWPTIPGEISWDVSFVTLNFLVPGLVIVISYSKILQTSEHLLDA
RAVVTHSEITKASRKRLTVSLAYSESHQIRVSQQDFRLFRTLFLLMVSFFIMWSPIIITI
LLILIQNFKQDLVIWPSLFFWVVAFTFANSALNPILYNMTLCRNEWKKIFCCFWFPEKGA
ILTDTSVKRNDLSIISG
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| BDBM382133 |
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| n/a |
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| Name | BDBM382133 |
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| Synonyms: | 4-(4-((2-(6-methoxypyridin-3-yl)cyclohex-1-en-1-yl)methoxy)phenyl) butanoic Acid | US10273230, Compound of Example 14 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H27NO4 |
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| Mol. Mass. | 381.4648 |
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| SMILES | COc1ccc(cn1)C1=C(COc2ccc(CCCC(O)=O)cc2)CCCC1 |c:9| |
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| Structure | 
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