Reaction Details |
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Target | Dual specificity protein phosphatase 6 |
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Ligand | BDBM31756 |
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Substrate/Competitor | 3-O-methylfluorescein phosphate (OMFP) |
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Meas. Tech. | In Vitro MKP-3 Dose Response Assay for SAR Study |
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pH | 7±n/a |
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Temperature | 296.15±n/a K |
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IC50 | 6000±n/a nM |
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Citation | PubChem, PC In Vitro MKP-3 Dose Response Assay for SAR Study PubChem Bioassay(2008)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Dual specificity protein phosphatase 6 |
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Name: | Dual specificity protein phosphatase 6 |
Synonyms: | DUS6_RAT | Dusp6 | MAP kinase phosphatase 3 | MKP-3 | Mitogen-activated protein kinase phosphatase 3 | Mkp3 |
Type: | Enzyme |
Mol. Mass.: | 42303.19 |
Organism: | Rattus norvegicus |
Description: | gi_16758752 |
Residue: | 381 |
Sequence: | MIDTLRPVPFASEMAISKTVAWLNEQLELGNEQLLLMDCRPQELYESSHIESAINVAIPG
IMLRRLQKGNLPVRALFTRCEDRDRFTRRCGTDTVVLYDENSSDWNENTGGESVLGLLLK
KLKDEGCRAFYLEGGFSKFQAEFALHCETNLDGSCSSSSPPLPVLGLGGLRISSDSSSDI
ESDLDRDPNSATDSDGSPLSNSQPSFPVEILPFLYLGCAKDSTNLDVLEEFGIKYILNVT
PNLPNLFENAGEFKYKQIPISDHWSQNLSQFFPEAISFIDEARGKNCGVLVHCLAGISRS
VTVTVAYLMQKLNLSMNDAYDIVKMKKSNISPNFNFMGQLLDFERTLGLSSPCDNRVPAQ
QLYFTAPSNQNVYQVDSLQST
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BDBM31756 |
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3-O-methylfluorescein phosphate (OMFP) |
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Name: | 3-O-methylfluorescein phosphate (OMFP) |
Synonyms: | n/a |
Type: | n/a |
Mol. Mass.: | 358.43 |
Organism: | n/a |
Description: | n/a |
Residue: | 3 |
Sequence: | |