| Reaction Details |
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 | Report a problem with these data |
| Target | Serine/threonine-protein kinase D1 |
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| Ligand | BDBM32350 |
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| Substrate/Competitor | Substrate Peptide |
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| Meas. Tech. | Fluorescence polarization assay for PKD inhibitiors-IC50 determinations |
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| pH | 7.2±n/a |
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| Temperature | 296.15±n/a K |
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| IC50 | >50000±n/a nM |
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| Citation |  PubChem, PC Fluorescence polarization assay for PKD inhibitiors-IC50 determinations PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Serine/threonine-protein kinase D1 |
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| Name: | Serine/threonine-protein kinase D1 |
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| Synonyms: | KPCD1_HUMAN | PKD | PKD1 | PRKCM | PRKD1 | Protein kinase C mu | Protein kinase C mu type | Protein kinase C mu type (PRKD1) | Protein kinase C, PKC; classical/novel | Protein kinase D | Protein kinase D (PRKD1) | Serine/threonine-protein kinase D1 (PKD1) | nPKC-D1 | nPKC-mu |
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| Type: | Serine/threonine-protein kinase |
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| Mol. Mass.: | 101705.07 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_115529463 |
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| Residue: | 912 |
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| Sequence: | MSAPPVLRPPSPLLPVAAAAAAAAAALVPGSGPGPAPFLAPVAAPVGGISFHLQIGLSRE
PVLLLQDSSGDYSLAHVREMACSIVDQKFPECGFYGMYDKILLFRHDPTSENILQLVKAA
SDIQEGDLIEVVLSASATFEDFQIRPHALFVHSYRAPAFCDHCGEMLWGLVRQGLKCEGC
GLNYHKRCAFKIPNNCSGVRRRRLSNVSLTGVSTIRTSSAELSTSAPDEPLLQKSPSESF
IGREKRSNSQSYIGRPIHLDKILMSKVKVPHTFVIHSYTRPTVCQYCKKLLKGLFRQGLQ
CKDCRFNCHKRCAPKVPNNCLGEVTINGDLLSPGAESDVVMEEGSDDNDSERNSGLMDDM
EEAMVQDAEMAMAECQNDSGEMQDPDPDHEDANRTISPSTSNNIPLMRVVQSVKHTKRKS
STVMKEGWMVHYTSKDTLRKRHYWRLDSKCITLFQNDTGSRYYKEIPLSEILSLEPVKTS
ALIPNGANPHCFEITTANVVYYVGENVVNPSSPSPNNSVLTSGVGADVARMWEIAIQHAL
MPVIPKGSSVGTGTNLHRDISVSISVSNCQIQENVDISTVYQIFPDEVLGSGQFGIVYGG
KHRKTGRDVAIKIIDKLRFPTKQESQLRNEVAILQNLHHPGVVNLECMFETPERVFVVME
KLHGDMLEMILSSEKGRLPEHITKFLITQILVALRHLHFKNIVHCDLKPENVLLASADPF
PQVKLCDFGFARIIGEKSFRRSVVGTPAYLAPEVLRNKGYNRSLDMWSVGVIIYVSLSGT
FPFNEDEDIHDQIQNAAFMYPPNPWKEISHEAIDLINNLLQVKMRKRYSVDKTLSHPWLQ
DYQTWLDLRELECKIGERYITHESDDLRWEKYAGEQGLQYPTHLINPSASHSDTPETEET
EMKALGERVSIL
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| BDBM32350 |
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| Substrate Peptide |
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| Name: | Substrate Peptide |
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| Synonyms: | n/a |
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| Type: | Peptide |
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| Mol. Mass.: | 358.43 |
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| Organism: | n/a |
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| Description: | ATP as co-substrate |
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| Residue: | 3 |
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| Sequence: | |
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