Reaction Details |
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Target | Dual specificity protein phosphatase 1 |
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Ligand | BDBM35379 |
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Substrate/Competitor | OMFP Substrate |
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Meas. Tech. | In vitro MKP-1 Phosphatase HTS Dose Response Confirmation Assay |
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pH | 7±n/a |
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Temperature | 295.15±n/a K |
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IC50 | 23124±n/a nM |
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Citation | PubChem, PC In vitro MKP-1 Phosphatase HTS Dose Response Confirmation Assay PubChem Bioassay(2007)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Dual specificity protein phosphatase 1 |
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Name: | Dual specificity protein phosphatase 1 |
Synonyms: | CL100 | DUS1_HUMAN | DUSP1 | Dual specificity protein phosphatase hVH1 | MAP kinase phosphatase 1 | MKP-1 | MKP1 | PTPN10 | Protein-tyrosine phosphatase CL100 | VH1 |
Type: | Protein phosphatase |
Mol. Mass.: | 39301.48 |
Organism: | Homo sapiens (Human) |
Description: | gi_4758204 |
Residue: | 367 |
Sequence: | MVMEVGTLDAGGLRALLGERAAQCLLLDCRSFFAFNAGHIAGSVNVRFSTIVRRRAKGAM
GLEHIVPNAELRGRLLAGAYHAVVLLDERSAALDGAKRDGTLALAAGALCREARAAQVFF
LKGGYEAFSASCPELCSKQSTPMGLSLPLSTSVPDSAESGCSSCSTPLYDQGGPVEILPF
LYLGSAYHASRKDMLDALGITALINVSANCPNHFEGHYQYKSIPVEDNHKADISSWFNEA
IDFIDSIKNAGGRVFVHCQAGISRSATICLAYLMRTNRVKLDEAFEFVKQRRSIISPNFS
FMGQLLQFESQVLAPHCSAEAGSPAMAVLDRGTSTTTVFNFPVSIPVHSTNSALSYLQSP
ITTSPSC
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BDBM35379 |
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OMFP Substrate |
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Name: | OMFP Substrate |
Synonyms: | 3-O-methylfluorescein phosphate | OMFP |
Type: | fluorescent substrate |
Mol. Mass.: | 358.43 |
Organism: | n/a |
Description: | n/a |
Residue: | 3 |
Sequence: | |