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TargetfMet-Leu-Phe receptor
LigandBDBM37643
Substrate/Competitorn/a
Meas. Tech.Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands
Ki 2200±n/a nM
Citation PubChem, PC Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands PubChem Bioassay(2007)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
fMet-Leu-Phe receptor
Name:fMet-Leu-Phe receptor
Synonyms:FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1
Type:Enzyme Catalytic Domain
Mol. Mass.:38456.14
Organism:Homo sapiens (Human)
Description:gi_4503779
Residue:350
Sequence:
METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
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BDBM37643
n/a
NameBDBM37643
Synonyms:(4Z)-5-(2,5-dimethoxyphenyl)-1-(2-furanylmethyl)-4-[hydroxy(phenyl)methylidene]pyrrolidine-2,3-dione | (4Z)-5-(2,5-dimethoxyphenyl)-1-(2-furfuryl)-4-[hydroxy(phenyl)methylene]pyrrolidine-2,3-quinone | (4Z)-5-(2,5-dimethoxyphenyl)-1-(furan-2-ylmethyl)-4-[hydroxy(phenyl)methylidene]pyrrolidine-2,3-dione | (4Z)-5-(2,5-dimethoxyphenyl)-1-(furan-2-ylmethyl)-4-[oxidanyl(phenyl)methylidene]pyrrolidine-2,3-dione | MLS000036525 | SMR000057915 | cid_5389251
TypeSmall organic molecule
Emp. Form.C24H21NO6
Mol. Mass.419.4266
SMILESCOc1ccc(OC)c(c1)C1C(C(=O)c2ccccc2)C(=O)C(=O)N1Cc1ccco1
Structure
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