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Reaction Details
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TargetfMet-Leu-Phe receptor
LigandBDBM37710
Substrate/Competitorn/a
Meas. Tech.Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands
Ki 16100±n/a nM
Citation PubChem, PC Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands PubChem Bioassay(2007)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
fMet-Leu-Phe receptor
Name:fMet-Leu-Phe receptor
Synonyms:FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1
Type:Enzyme Catalytic Domain
Mol. Mass.:38456.14
Organism:Homo sapiens (Human)
Description:gi_4503779
Residue:350
Sequence:
METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
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  Blast E-value cutoff:
BDBM37710
n/a
NameBDBM37710
Synonyms:(4Z)-4-[hydroxy(phenyl)methylene]-1-(2-hydroxypropyl)-5-(2-methoxyphenyl)pyrrolidine-2,3-quinone | (4Z)-4-[hydroxy(phenyl)methylidene]-1-(2-hydroxypropyl)-5-(2-methoxyphenyl)pyrrolidine-2,3-dione | (4Z)-5-(2-methoxyphenyl)-4-[oxidanyl(phenyl)methylidene]-1-(2-oxidanylpropyl)pyrrolidine-2,3-dione | 4-benzoyl-3-hydroxy-1-(2-hydroxypropyl)-5-(2-methoxyphenyl)-1,5-dihydro-2H-pyrrol-2-one | MLS000090218 | SMR000024829 | cid_5771369
TypeSmall organic molecule
Emp. Form.C21H21NO5
Mol. Mass.367.3951
SMILESCOc1ccccc1C1C(C(=O)c2ccccc2)C(=O)C(=O)N1CC(C)O
Structure
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