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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | fMet-Leu-Phe receptor | ||
| Ligand | BDBM34503 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands | ||
| Ki | 12900±n/a nM | ||
| Citation |  PubChem, PC Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands PubChem Bioassay(2007)[AID] | ||
| More Info.: | Get all data from this article, Solution Info, Assay Method | ||
| fMet-Leu-Phe receptor | |||
| Name: | fMet-Leu-Phe receptor | ||
| Synonyms: | FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1 | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 38456.14 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | gi_4503779 | ||
| Residue: | 350 | ||
| Sequence: |
| ||
| BDBM34503 | |||
| n/a | |||
| Name | BDBM34503 | ||
| Synonyms: | 3-cyclohexyl-6-keto-8-(2-methoxy-1-naphthyl)-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile | 3-cyclohexyl-8-(2-methoxy-1-naphthalenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile | 3-cyclohexyl-8-(2-methoxynaphthalen-1-yl)-6-oxidanylidene-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile | 3-cyclohexyl-8-(2-methoxynaphthalen-1-yl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile | MLS000117271 | SMR000094223 | cid_5307697 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C25H27N3O2S | ||
| Mol. Mass. | 433.566 | ||
| SMILES | COc1ccc2ccccc2c1C1CC(=O)N2CN(CSC2=C1C#N)C1CCCCC1 |c:24| | ||
| Structure | 
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