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TargetfMet-Leu-Phe receptor
LigandBDBM37824
Substrate/Competitorn/a
Meas. Tech.Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands
Ki 7500±n/a nM
Citation PubChem, PC Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands PubChem Bioassay(2007)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
fMet-Leu-Phe receptor
Name:fMet-Leu-Phe receptor
Synonyms:FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1
Type:Enzyme Catalytic Domain
Mol. Mass.:38456.14
Organism:Homo sapiens (Human)
Description:gi_4503779
Residue:350
Sequence:
METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
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  Blast E-value cutoff:
BDBM37824
n/a
NameBDBM37824
Synonyms:4-(1-adamantyl)-1,2-diphenyl-pyrazolidine-3,5-dione | 4-(1-adamantyl)-1,2-diphenyl-pyrazolidine-3,5-quinone | 4-(1-adamantyl)-1,2-diphenylpyrazolidine-3,5-dione | 4-Adamantan-1-yl-1,2-diphenyl-pyrazolidine-3,5-dione | MLS000526352 | SMR000116826 | cid_2831216
TypeSmall organic molecule
Emp. Form.C25H26N2O2
Mol. Mass.386.4861
SMILES[H]C12CC3([H])CC([H])(C1)CC(C2)(C3)c1c(O)n(-c2ccccc2)n(-c2ccccc2)c1=O |TLB:8:1:12:6.9.5,8:6:12:1.11.2,THB:2:1:9:3.12.5,2:3:9:1.11.8|
Structure
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