| Reaction Details |
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 | Report a problem with these data |
| Target | cAMP-dependent protein kinase catalytic subunit alpha |
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| Ligand | BDBM37913 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose-response biochemical assay for inhibitors of protein kinase A (PKA) activity |
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| IC50 | 1761±n/a nM |
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| Citation |  PubChem, PC Dose-response biochemical assay for inhibitors of protein kinase A (PKA) activity PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| cAMP-dependent protein kinase catalytic subunit alpha |
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| Name: | cAMP-dependent protein kinase catalytic subunit alpha |
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| Synonyms: | KAPCA_HUMAN | PKA C-alpha | PKACA | PRKACA | cAMP-dependent protein kinase (PKA) | cAMP-dependent protein kinase catalytic (PKA) | cAMP-dependent protein kinase catalytic subunit alpha | cAMP-dependent protein kinase catalytic subunit alpha (PKA) | cAMP-dependent protein kinase catalytic subunit alpha (PKACA) | cAMP-dependent protein kinase catalytic subunit alpha (PKAc) | cAMP-dependent protein kinase catalytic subunit alpha isoform 1 | cAMP-dependent protein kinase, alpha-catalytic subunit |
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| Type: | Enzyme Catalytic Subunit |
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| Mol. Mass.: | 40598.73 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 351 |
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| Sequence: | MGNAAAAKKGSEQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVML
VKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMV
MEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGY
IQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFF
ADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFAT
TDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF
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| BDBM37913 |
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| n/a |
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| Name | BDBM37913 |
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| Synonyms: | MLS000065710 | N-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)-2-thiophen-2-yl-ethanamide | N-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)-2-thiophen-2-ylacetamide | N-[5-(4-pyridinyl)-1,3,4-thiadiazol-2-yl]-2-(2-thienyl)acetamide | N-[5-(4-pyridyl)-1,3,4-thiadiazol-2-yl]-2-(2-thienyl)acetamide | SMR000080373 | cid_1245524 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H10N4OS2 |
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| Mol. Mass. | 302.375 |
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| SMILES | O=C(Cc1cccs1)Nc1nnc(s1)-c1ccncc1 |
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| Structure | 
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