Ki Summary

Reaction Details

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Target

Dual specificity protein phosphatase 6

Ligand

BDBM35386

Substrate/Competitor

n/a

Meas. Tech.

In vitro MKP-3 Phosphatase Dose Response Active/Probe Assessment Assay - Reproducibility testing

IC50

>50000±n/a nM

Citation

PubChem, PC In vitro MKP-3 Phosphatase Dose Response Active/Probe Assessment Assay - Reproducibility testing PubChem Bioassay(2007)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Dual specificity protein phosphatase 6

Name:

Dual specificity protein phosphatase 6

Synonyms:

Type:

Enzyme

Mol. Mass.:

42303.19

Organism:

Rattus norvegicus

Description:

gi_16758752

Residue:

381

Sequence:

MIDTLRPVPFASEMAISKTVAWLNEQLELGNEQLLLMDCRPQELYESSHIESAINVAIPG
IMLRRLQKGNLPVRALFTRCEDRDRFTRRCGTDTVVLYDENSSDWNENTGGESVLGLLLK
KLKDEGCRAFYLEGGFSKFQAEFALHCETNLDGSCSSSSPPLPVLGLGGLRISSDSSSDI
ESDLDRDPNSATDSDGSPLSNSQPSFPVEILPFLYLGCAKDSTNLDVLEEFGIKYILNVT
PNLPNLFENAGEFKYKQIPISDHWSQNLSQFFPEAISFIDEARGKNCGVLVHCLAGISRS
VTVTVAYLMQKLNLSMNDAYDIVKMKKSNISPNFNFMGQLLDFERTLGLSSPCDNRVPAQ
QLYFTAPSNQNVYQVDSLQST

BDBM35386

n/a

Name

BDBM35386

Synonyms:

MLS000095236 | N-(4-ethylphenyl)-2-[3-(2-morpholin-4-ylethyl)-4-oxidanylidene-quinazolin-2-yl]sulfanyl-ethanamide | N-(4-ethylphenyl)-2-[3-(2-morpholin-4-ylethyl)-4-oxoquinazolin-2-yl]sulfanylacetamide | N-(4-ethylphenyl)-2-[[3-[2-(4-morpholinyl)ethyl]-4-oxo-2-quinazolinyl]thio]acetamide | N-(4-ethylphenyl)-2-[[4-keto-3-(2-morpholinoethyl)quinazolin-2-yl]thio]acetamide | N-(4-ethylphenyl)-2-{[3-(2-morpholin-4-ylethyl)-4-oxo-3,4-dihydroquinazolin-2-yl]thio}acetamide | SMR000030790 | cid_3237221

Type

Small organic molecule

Emp. Form.

C24H28N4O3S

Mol. Mass.

452.569

SMILES

CCc1ccc(NC(=O)CSc2nc3ccccc3c(=O)n2CCN2CCOCC2)cc1

Structure