Reaction Details |
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Target | Isoform 2 of Nuclear receptor ROR-alpha (Alpha-2) |
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Ligand | BDBM38994 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose-response cell-based assay for inhibitors of the Retinoic Acid Receptor-related orphan receptor A (RORA) |
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IC50 | 727±n/a nM |
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Citation | PubChem, PC Dose-response cell-based assay for inhibitors of the Retinoic Acid Receptor-related orphan receptor A (RORA) PubChem Bioassay(2007)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Isoform 2 of Nuclear receptor ROR-alpha (Alpha-2) |
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Name: | Isoform 2 of Nuclear receptor ROR-alpha (Alpha-2) |
Synonyms: | NR1F1 | Nuclear receptor ROR-alpha | Nuclear receptor ROR-alpha (Alpha-2) | Nuclear receptor ROR-alpha (Retinoid-related orphan receptor-alpha) (Nuclear receptor RZR-alpha). | RORA | RORA_HUMAN | RZRA |
Type: | PROTEIN |
Mol. Mass.: | 63033.59 |
Organism: | Homo sapiens (Human) |
Description: | EBI_101591 |
Residue: | 556 |
Sequence: | MNEGAPGDSDLETEARVPWSIMGHCLRTGQARMSATPTPAGEGARRDELFGILQILHQCI
LSSGDAFVLTGVCCSWRQNGKPPYSQKEDKEVQTGYMNAQIEIIPCKICGDKSSGIHYGV
ITCEGCKGFFRRSQQSNATYSCPRQKNCLIDRTSRNRCQHCRLQKCLAVGMSRDAVKFGR
MSKKQRDSLYAEVQKHRMQQQQRDHQQQPGEAEPLTPTYNISANGLTELHDDLSNYIDGH
TPEGSKADSAVSSFYLDIQPSPDQSGLDINGIKPEPICDYTPASGFFPYCSFTNGETSPT
VSMAELEHLAQNISKSHLETCQYLREELQQITWQTFLQEEIENYQNKQREVMWQLCAIKI
TEAIQYVVEFAKRIDGFMELCQNDQIVLLKAGSLEVVFIRMCRAFDSQNNTVYFDGKYAS
PDVFKSLGCEDFISFVFEFGKSLCSMHLTEDEIALFSAFVLMSADRSWLQEKVKIEKLQQ
KIQLALQHVLQKNHREDGILTKLICKVSTLRALCGRHTEKLMAFKAIYPDIVRLHFPPLY
KELFTSEFEPAMQIDG
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BDBM38994 |
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n/a |
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Name | BDBM38994 |
Synonyms: | MLS000089367 | N-(2-methoxyethyl)-2-[({5-methyl-2-[4-(methylthio)phenyl]-1,3-oxazol-4-yl}methyl)thio]acetamide | N-(2-methoxyethyl)-2-[[5-methyl-2-(4-methylsulfanylphenyl)-1,3-oxazol-4-yl]methylsulfanyl]acetamide | N-(2-methoxyethyl)-2-[[5-methyl-2-(4-methylsulfanylphenyl)-1,3-oxazol-4-yl]methylsulfanyl]ethanamide | N-(2-methoxyethyl)-2-[[5-methyl-2-[4-(methylthio)phenyl]-4-oxazolyl]methylthio]acetamide | N-(2-methoxyethyl)-2-[[5-methyl-2-[4-(methylthio)phenyl]oxazol-4-yl]methylthio]acetamide | SMR000027742 | cid_3245395 |
Type | Small organic molecule |
Emp. Form. | C17H22N2O3S2 |
Mol. Mass. | 366.498 |
SMILES | COCCNC(=O)CSCc1nc(oc1C)-c1ccc(SC)cc1 |
Structure |
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