| Reaction Details |
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 | Report a problem with these data |
| Target | Steroidogenic factor 1 |
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| Ligand | BDBM38845 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Counterscreen for inhibitors of the Retinoic Acid Receptor-related orphan receptor A (RORA): A cell-based dose-response assay for inhibition of the Steroidogenic Factor 1 (SF-1) |
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| IC50 | 7643±n/a nM |
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| Citation |  PubChem, PC Counterscreen for inhibitors of the Retinoic Acid Receptor-related orphan receptor A (RORA): A cell-based dose-response assay for inhibition of the Steroidogenic Factor 1 (SF-1) PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Steroidogenic factor 1 |
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| Name: | Steroidogenic factor 1 |
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| Synonyms: | AD4BP | Adrenal 4-binding protein | FTZF1 | Fushi tarazu factor homolog 1 | NR5A1 | Nuclear receptor subfamily 5 group A member 1 | SF-1 | SF1 | STF-1 | STF1_HUMAN | Steroid hormone receptor Ad4BP |
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| Type: | Nuclear Hormone Receptor |
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| Mol. Mass.: | 51643.43 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 461 |
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| Sequence: | MDYSYDEDLDELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKHYTCTESQSCKIDKT
QRKRCPFCRFQKCLTVGMRLEAVRADRMRGGRNKFGPMYKRDRALKQQKKAQIRANGFKL
ETGPPMGVPPPPPPAPDYVLPPSLHGPEPKGLAAGPPAGPLGDFGAPALPMAVPGAHGPL
AGYLYPAFPGRAIKSEYPEPYASPPQPGLPYGYPEPFSGGPNVPELILQLLQLEPDEDQV
RARILGCLQEPTKSRPDQPAAFGLLCRMADQTFISIVDWARRCMVFKELEVADQMTLLQN
CWSELLVFDHIYRQVQHGKEGSILLVTGQEVELTTVATQAGSLLHSLVLRAQELVLQLLA
LQLDRQEFVCLKFIILFSLDLKFLNNHILVKDAQEKANAALLDYTLCHYPHCGDKFQQLL
LCLVEVRALSMQAKEYLYHKHLGNEMPRNNLLIEMLQAKQT
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| BDBM38845 |
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| n/a |
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| Name | BDBM38845 |
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| Synonyms: | MLS000032332 | N-[4-(2-{5-[(4-Chloro-phenylamino)-methyl]-[1,3,4]oxadiazol-2-ylsulfanyl}-acetyl)-2-ethoxy-phenyl]-propionamide | N-[4-[2-[[5-[(4-chloroanilino)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]-2-ethoxyphenyl]propanamide | N-[4-[2-[[5-[(4-chloroanilino)methyl]-1,3,4-oxadiazol-2-yl]thio]-1-oxoethyl]-2-ethoxyphenyl]propanamide | N-[4-[2-[[5-[(4-chloroanilino)methyl]-1,3,4-oxadiazol-2-yl]thio]acetyl]-2-ethoxy-phenyl]propionamide | N-[4-[2-[[5-[[(4-chlorophenyl)amino]methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethanoyl]-2-ethoxy-phenyl]propanamide | SMR000003314 | cid_644459 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H23ClN4O4S |
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| Mol. Mass. | 474.96 |
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| SMILES | CCOc1cc(ccc1NC(=O)CC)C(=O)CSc1nnc(CNc2ccc(Cl)cc2)o1 |
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| Structure | 
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