| Reaction Details |
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 | Report a problem with these data |
| Target | Isoform 2 of Nuclear receptor ROR-alpha (Alpha-2) |
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| Ligand | BDBM39467 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Counterscreen for activators of the nuclear receptor Steroidogenic Factor 1 (SF-1): A cell-based dose-response assay for inhibition of the RAR-related orphan receptor A (RORA) |
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| EC50 | 897±n/a nM |
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| Citation |  PubChem, PC Counterscreen for activators of the nuclear receptor Steroidogenic Factor 1 (SF-1): A cell-based dose-response assay for inhibition of the RAR-related orphan receptor A (RORA) PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Isoform 2 of Nuclear receptor ROR-alpha (Alpha-2) |
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| Name: | Isoform 2 of Nuclear receptor ROR-alpha (Alpha-2) |
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| Synonyms: | NR1F1 | Nuclear receptor ROR-alpha | Nuclear receptor ROR-alpha (Alpha-2) | Nuclear receptor ROR-alpha (Retinoid-related orphan receptor-alpha) (Nuclear receptor RZR-alpha). | RORA | RORA_HUMAN | RZRA |
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| Type: | PROTEIN |
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| Mol. Mass.: | 63033.59 |
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| Organism: | Homo sapiens (Human) |
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| Description: | EBI_101591 |
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| Residue: | 556 |
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| Sequence: | MNEGAPGDSDLETEARVPWSIMGHCLRTGQARMSATPTPAGEGARRDELFGILQILHQCI
LSSGDAFVLTGVCCSWRQNGKPPYSQKEDKEVQTGYMNAQIEIIPCKICGDKSSGIHYGV
ITCEGCKGFFRRSQQSNATYSCPRQKNCLIDRTSRNRCQHCRLQKCLAVGMSRDAVKFGR
MSKKQRDSLYAEVQKHRMQQQQRDHQQQPGEAEPLTPTYNISANGLTELHDDLSNYIDGH
TPEGSKADSAVSSFYLDIQPSPDQSGLDINGIKPEPICDYTPASGFFPYCSFTNGETSPT
VSMAELEHLAQNISKSHLETCQYLREELQQITWQTFLQEEIENYQNKQREVMWQLCAIKI
TEAIQYVVEFAKRIDGFMELCQNDQIVLLKAGSLEVVFIRMCRAFDSQNNTVYFDGKYAS
PDVFKSLGCEDFISFVFEFGKSLCSMHLTEDEIALFSAFVLMSADRSWLQEKVKIEKLQQ
KIQLALQHVLQKNHREDGILTKLICKVSTLRALCGRHTEKLMAFKAIYPDIVRLHFPPLY
KELFTSEFEPAMQIDG
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| BDBM39467 |
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| n/a |
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| Name | BDBM39467 |
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| Synonyms: | 2,5-dimethyl-3-furancarboxylic acid [2-(2,3-dihydroindol-1-yl)-2-oxoethyl] ester | 2,5-dimethylfuran-3-carboxylic acid (2-indolin-1-yl-2-keto-ethyl) ester | MLS000097673 | SMR000061688 | [2-(2,3-dihydroindol-1-yl)-2-oxidanylidene-ethyl] 2,5-dimethylfuran-3-carboxylate | [2-(2,3-dihydroindol-1-yl)-2-oxoethyl] 2,5-dimethylfuran-3-carboxylate | cid_2369751 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H17NO4 |
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| Mol. Mass. | 299.3212 |
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| SMILES | Cc1cc(C(=O)OCC(=O)N2CCc3ccccc23)c(C)o1 |
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| Structure | 
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