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Target14-3-3 protein gamma
LigandBDBM39864
Substrate/Competitorn/a
Meas. Tech.14-3-3 protein interaction modulators Dose Response Confirmation
IC50 29952.3±n/a nM
Citation PubChem, PC 14-3-3 protein interaction modulators Dose Response Confirmation PubChem Bioassay(2007)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
14-3-3 protein gamma
Name:14-3-3 protein gamma
Synonyms:1433G_HUMAN | YWHAG | tyrosine 3-monooxygenase/tryptophan 5-monooxygenase activation protein, gamma polypeptide
Type:Enzyme Catalytic Domain
Mol. Mass.:28289.17
Organism:Homo sapiens (Human)
Description:gi_21464101
Residue:247
Sequence:
MVDREQLVQKARLAEQAERYDDMAAAMKNVTELNEPLSNEERNLLSVAYKNVVGARRSSW
RVISSIEQKTSADGNEKKIEMVRAYREKIEKELEAVCQDVLSLLDNYLIKNCSETQYESK
VFYLKMKGDYYRYLAEVATGEKRATVVESSEKAYSEAHEISKEHMQPTHPIRLGLALNYS
VFYYEIQNAPEQACHLAKTAFDDAIAELDTLNEDSYKDSTLIMQLLRDNLTLWTSDQQDD
DGGEGNN
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  Blast E-value cutoff:
BDBM39864
n/a
NameBDBM39864
Synonyms:(4-methoxy-7,7-dimethyl-6,8-dihydropyrimido[4,5-b][1,4]benzothiazin-9-yl)amine;hydrobromide | 4-methoxy-7,7-dimethyl-6,8-dihydropyrimido[4,5-b][1,4]benzothiazin-9-amine;hydrobromide | MLS000038875 | SMR000036340 | cid_6602809
TypeSmall organic molecule
Emp. Form.C13H16N4OS
Mol. Mass.276.357
SMILESCOc1ncnc2SC3=C(N)CC(C)(C)CC3=Nc12 |c:8,17|
Structure
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