| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Ubiquitin carboxyl-terminal hydrolase BAP1 |
|---|
| Ligand | BDBM40276 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | BAP1 Enzyme inhibitors Dose Response Confirmation |
|---|
| IC50 | 23100.9±n/a nM |
|---|
| Citation |  PubChem, PC BAP1 Enzyme inhibitors Dose Response Confirmation PubChem Bioassay(2007)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Ubiquitin carboxyl-terminal hydrolase BAP1 |
|---|
| Name: | Ubiquitin carboxyl-terminal hydrolase BAP1 |
|---|
| Synonyms: | BAP1 | BAP1_HUMAN | KIAA0272 | Ubiquitin carboxyl-terminal hydrolase BAP1 (BRCA1-associated protein 1) (Cerebral protein 6). |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 80364.15 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_68565074 |
|---|
| Residue: | 729 |
|---|
| Sequence: | MNKGWLELESDPGLFTLLVEDFGVKGVQVEEIYDLQSKCQGPVYGFIFLFKWIEERRSRR
KVSTLVDDTSVIDDDIVNNMFFAHQLIPNSCATHALLSVLLNCSSVDLGPTLSRMKDFTK
GFSPESKGYAIGNAPELAKAHNSHARPEPRHLPEKQNGLSAVRTMEAFHFVSYVPITGRL
FELDGLKVYPIDHGPWGEDEEWTDKARRVIMERIGLATAGEPYHDIRFNLMAVVPDRRIK
YEARLHVLKVNRQTVLEALQQLIRVTQPELIQTHKSQESQLPEESKSASNKSPLVLEANR
APAASEGNHTDGAEEAAGSCAQAPSHSPPNKPKLVVKPPGSSLNGVHPNPTPIVQRLPAF
LDNHNYAKSPMQEEEDLAAGVGRSRVPVRPPQQYSDDEDDYEDDEEDDVQNTNSALRYKG
KGTGKPGALSGSADGQLSVLQPNTINVLAEKLKESQKDLSIPLSIKTSSGAGSPAVAVPT
HSQPSPTPSNESTDTASEIGSAFNSPLRSPIRSANPTRPSSPVTSHISKVLFGEDDSLLR
VDCIRYNRAVRDLGPVISTGLLHLAEDGVLSPLALTEGGKGSSPSIRPIQGSQGSSSPVE
KEVVEATDSREKTGMVRPGEPLSGEKYSPKELLALLKCVEAEIANYEACLKEEVEKRKKF
KIDDQRRTHNYDEFICTFISMLAQEGMLANLVEQNISVRRRQGVSIGRLHKQRKPDRRKR
SRPYKAKRQ
|
|
|
|---|
| BDBM40276 |
|---|
| n/a |
|---|
| Name | BDBM40276 |
|---|
| Synonyms: | 5-Acetyl-4-methyl-2-[2-(5-phenyl-tetrazol-2-yl)-acetylamino]-thiophene-3-carboxylic acid ethyl ester | 5-acetyl-4-methyl-2-[[1-oxo-2-(5-phenyl-2-tetrazolyl)ethyl]amino]-3-thiophenecarboxylic acid ethyl ester | 5-acetyl-4-methyl-2-[[2-(5-phenyltetrazol-2-yl)acetyl]amino]thiophene-3-carboxylic acid ethyl ester | MLS000071676 | SMR000001564 | cid_651347 | ethyl 5-acetyl-4-methyl-2-[[2-(5-phenyltetrazol-2-yl)acetyl]amino]thiophene-3-carboxylate | ethyl 5-ethanoyl-4-methyl-2-[2-(5-phenyl-1,2,3,4-tetrazol-2-yl)ethanoylamino]thiophene-3-carboxylate |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H19N5O4S |
|---|
| Mol. Mass. | 413.45 |
|---|
| SMILES | CCOC(=O)c1c(C)c(sc1NC(=O)Cn1nnc(n1)-c1ccccc1)C(C)=O |
|---|
| Structure | 
|
|---|
Search and Browse
