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Reaction Details
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TargetN-formyl peptide receptor 2
LigandBDBM40420
Substrate/Competitorn/a
Meas. Tech.Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay Counterscreen Against Formyl Peptide Receptor-Like-1 (FPRL1)
Ki>40300±n/a nM
Citation PubChem, PC Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay Counterscreen Against Formyl Peptide Receptor-Like-1 (FPRL1)  PubChem Bioassay(2007)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
N-formyl peptide receptor 2
Name:N-formyl peptide receptor 2
Synonyms:ALXR, FPRL1, FPR2 | FMLP-related receptor I FMLP-R-I | FPR2 | FPR2_HUMAN | FPRH1 | FPRL1 | Formyl Peptide Receptor-Like 1 | HM63 | LXA4 receptor | LXA4R | Lipoxin A4 receptor | Lipoxin A4 receptor (LXA4) | RFP | hFPRL
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:38968.35
Organism:Homo sapiens (Human)
Description:P25090
Residue:351
Sequence:
METNFSTPLNEYEEVSYESAGYTVLRILPLVVLGVTFVLGVLGNGLVIWVAGFRMTRTVT
TICYLNLALADFSFTATLPFLIVSMAMGEKWPFGWFLCKLIHIVVDINLFGSVFLIGFIA
LDRCICVLHPVWAQNHRTVSLAMKVIVGPWILALVLTLPVFLFLTTVTIPNGDTYCTFNF
ASWGGTPEERLKVAITMLTARGIIRFVIGFSLPMSIVAICYGLIAAKIHKKGMIKSSRPL
RVLTAVVASFFICWFPFQLVALLGTVWLKEMLFYGKYKIIDILVNPTSSLAFFNSCLNPM
LYVFVGQDFRERLIHSLPTSLERALSEDSAPTNDTAANSASPPAETELQAM
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  Blast E-value cutoff:
BDBM40420
n/a
NameBDBM40420
Synonyms:1-(3-imidazol-1-ylpropyl)-2-(4-methoxyphenyl)-4-oxidanyl-3-thiophen-2-ylcarbonyl-2H-pyrrol-5-one | 3-hydroxy-1-(3-imidazol-1-ylpropyl)-5-(4-methoxyphenyl)-4-(2-thenoyl)-3-pyrrolin-2-one | 4-hydroxy-1-(3-imidazol-1-ylpropyl)-2-(4-methoxyphenyl)-3-(thiophene-2-carbonyl)-2H-pyrrol-5-one | 4-hydroxy-1-[3-(1-imidazolyl)propyl]-2-(4-methoxyphenyl)-3-[oxo(thiophen-2-yl)methyl]-2H-pyrrol-5-one | UNM000003552401 | cid_2907867
TypeSmall organic molecule
Emp. Form.C22H21N3O4S
Mol. Mass.423.485
SMILESCOc1ccc(cc1)C1C(C(=O)c2cccs2)C(=O)C(=O)N1CCCn1ccnc1
Structure
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