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TargetNuclear receptor subfamily 4 group A member 1
LigandBDBM40571
Substrate/Competitorn/a
Meas. Tech.High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters
IC50>12500±0 nM
Citation PubChem, PC High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Nuclear receptor subfamily 4 group A member 1
Name:Nuclear receptor subfamily 4 group A member 1
Synonyms:GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1
Type:Enzyme Catalytic Domain
Mol. Mass.:64467.13
Organism:Homo sapiens (Human)
Description:gi_27894344
Residue:598
Sequence:
MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM40571
n/a
NameBDBM40571
Synonyms:3-amino-6-methyl-7-thiazolo[3,2-b][1,2,4]triazinone | 3-amino-6-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazin-7-one | 3-amino-6-methyl-thiazolo[3,2-b][1,2,4]triazin-7-one | 3-azanyl-6-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazin-7-one | MLS000032547 | SMR000012776 | cid_648831
TypeSmall organic molecule
Emp. Form.C6H6N4OS
Mol. Mass.182.203
SMILESCc1nn2c(N)csc2nc1=O
Structure
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