Ki Summary

Reaction Details

Report a problem with these data

Target

Nuclear receptor subfamily 4 group A member 1

Ligand

BDBM40577

Substrate/Competitor

n/a

Meas. Tech.

High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters

IC50

43912±1230 nM

Citation

PubChem, PC High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters PubChem Bioassay(2008)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Nuclear receptor subfamily 4 group A member 1

Name:

Nuclear receptor subfamily 4 group A member 1

Synonyms:

GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1

Type:

Enzyme Catalytic Domain

Mol. Mass.:

64467.13

Organism:

Homo sapiens (Human)

Description:

gi_27894344

Residue:

598

Sequence:

MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF

BDBM40577

n/a

Name

BDBM40577

Synonyms:

4-(4-Pyrrolidin-1-yl-quinazolin-2-ylamino)-phenol | 4-[(4-pyrrolidin-1-ylquinazolin-2-yl)amino]phenol;hydrochloride | 4-[(4-pyrrolidinoquinazolin-2-yl)amino]phenol;hydrochloride | 4-[[4-(1-pyrrolidinyl)-2-quinazolinyl]amino]phenol;hydrochloride | MLS000026828 | SMR000013024 | cid_6602552

Type

Small organic molecule

Emp. Form.

C18H18N4O

Mol. Mass.

306.3617

SMILES

Oc1ccc(Nc2nc(N3CCCC3)c3ccccc3n2)cc1

Structure