| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Nuclear receptor subfamily 4 group A member 1 |
|---|
| Ligand | BDBM40591 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters |
|---|
| IC50 | >12500±0 nM |
|---|
| Citation |  PubChem, PC High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters PubChem Bioassay(2008)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Nuclear receptor subfamily 4 group A member 1 |
|---|
| Name: | Nuclear receptor subfamily 4 group A member 1 |
|---|
| Synonyms: | GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 64467.13 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_27894344 |
|---|
| Residue: | 598 |
|---|
| Sequence: | MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF
|
|
|
|---|
| BDBM40591 |
|---|
| n/a |
|---|
| Name | BDBM40591 |
|---|
| Synonyms: | 2-azanylidene-1-methyl-3-(phenylsulfonyl)dipyrido[1,2-e:4',3'-f]pyrimidin-5-one | 3-(benzenesulfonyl)-2-imino-1-methyl-5-dipyrido[1,2-e:4',3'-f]pyrimidinone | 3-(benzenesulfonyl)-2-imino-1-methyldipyrido[1,2-e:4',3'-f]pyrimidin-5-one | 3-besyl-2-imino-1-methyl-dipyrido[1,2-e:4',3'-f]pyrimidin-5-one | MLS000078666 | SMR000041828 | cid_661265 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C18H14N4O3S |
|---|
| Mol. Mass. | 366.394 |
|---|
| SMILES | Cn1c2nc3ccccn3c(=O)c2cc(c1=N)S(=O)(=O)c1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
