Ki Summary

Reaction Details

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Target

Nuclear receptor subfamily 4 group A member 1

Ligand

BDBM40622

Substrate/Competitor

n/a

Meas. Tech.

High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters

IC50

16351±1180 nM

Citation

PubChem, PC High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters PubChem Bioassay(2008)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Nuclear receptor subfamily 4 group A member 1

Name:

Nuclear receptor subfamily 4 group A member 1

Synonyms:

GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1

Type:

Enzyme Catalytic Domain

Mol. Mass.:

64467.13

Organism:

Homo sapiens (Human)

Description:

gi_27894344

Residue:

598

Sequence:

MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF

BDBM40622

n/a

Name

BDBM40622

Synonyms:

MLS000053340 | N-(2-furanylmethyl)-2,3-dihydro-1H-cyclopenta[b]quinoline-9-carboxamide | N-(2-furfuryl)-2,3-dihydro-1H-cyclopenta[b]quinoline-9-carboxamide | N-(furan-2-ylmethyl)-2,3-dihydro-1H-cyclopenta[b]quinoline-9-carboxamide | SMR000067677 | cid_862194

Type

Small organic molecule

Emp. Form.

C18H16N2O2

Mol. Mass.

292.3318

SMILES

O=C(NCc1ccco1)c1c2CCCc2nc2ccccc12

Structure