| Reaction Details |
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 | Report a problem with these data |
| Target | fMet-Leu-Phe receptor |
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| Ligand | BDBM40749 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Formylpeptide Receptor (FPRL1) Ligand Structure Activity Relationship (SAR) Analysis : FPR Dose Response Counterscreen Assay |
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| IC50 | >75000±n/a nM |
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| Citation |  PubChem, PC Formylpeptide Receptor (FPRL1) Ligand Structure Activity Relationship (SAR) Analysis : FPR Dose Response Counterscreen Assay PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| fMet-Leu-Phe receptor |
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| Name: | fMet-Leu-Phe receptor |
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| Synonyms: | FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 38456.14 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_4503779 |
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| Residue: | 350 |
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| Sequence: | METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
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| BDBM40749 |
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| n/a |
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| Name | BDBM40749 |
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| Synonyms: | N-(5-imidazo[1,2-a]pyrimidin-2-yl-2-methoxy-phenyl)propanamide | N-(5-imidazo[1,2-a]pyrimidin-2-yl-2-methoxy-phenyl)propionamide | N-(5-imidazo[1,2-a]pyrimidin-2-yl-2-methoxyphenyl)propanamide | N-[5-(2-imidazo[1,2-a]pyrimidinyl)-2-methoxyphenyl]propanamide | UNM000003657601 | cid_7080248 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H16N4O2 |
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| Mol. Mass. | 296.3238 |
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| SMILES | CCC(=O)Nc1cc(ccc1OC)-c1cn2cccnc2n1 |
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| Structure | 
|
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