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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Cathepsin B | ||
| Ligand | BDBM32102 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Cathepsin B dose-response confirmation | ||
| IC50 | 46.1±2.6 nM | ||
| Citation |  PubChem, PC Cathepsin B dose-response confirmation PubChem Bioassay(2008)[AID] | ||
| More Info.: | Get all data from this article, Solution Info, Assay Method | ||
| Cathepsin B | |||
| Name: | Cathepsin B | ||
| Synonyms: | APP secretase | APPS | CATB_HUMAN | CPSB | CTSB | Cathepsin B heavy chain | Cathepsin B light chain | Cathepsin B1 | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 37819.69 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | gi_63102437 | ||
| Residue: | 339 | ||
| Sequence: |
| ||
| BDBM32102 | |||
| n/a | |||
| Name | BDBM32102 | ||
| Synonyms: | 1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,6H)-dione | 1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | 1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7-quinone | MLS000087831 | SMR000024051 | US9284299, PKF118-310 | US9738628, Compound PKF118-310 | cid_66541 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C7H7N5O2 | ||
| Mol. Mass. | 193.1628 | ||
| SMILES | Cn1ncnc2c1nc(=O)n(C)c2=O | ||
| Structure | 
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