Ki Summary

Reaction Details

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Target

Sphingosine 1-phosphate receptor 2

Ligand

BDBM41668

Substrate/Competitor

n/a

Meas. Tech.

Dose Response Cell Based Assay for Agonists of the S1P2 Receptor

EC50

4549±n/a nM

Citation

PubChem, PC Dose Response Cell Based Assay for Agonists of the S1P2 Receptor PubChem Bioassay(2007)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Sphingosine 1-phosphate receptor 2

Name:

Sphingosine 1-phosphate receptor 2

Synonyms:

Type:

G Protein-Coupled Receptor (GPCR)

Mol. Mass.:

38883.16

Organism:

Homo sapiens (Human)

Description:

Membranes isolated from S1P2-transfected CHO cells were used in ligand binding assay.

Residue:

353

Sequence:

MGSLYSEYLNPNKVQEHYNYTKETLETQETTSRQVASAFIVILCCAIVVENLLVLIAVAR
NSKFHSAMYLFLGNLAASDLLAGVAFVANTLLSGSVTLRLTPVQWFAREGSAFITLSASV
FSLLAIAIERHVAIAKVKLYGSDKSCRMLLLIGASWLISLVLGGLPILGWNCLGHLEACS
TVLPLYAKHYVLCVVTIFSIILLAIVALYVRIYCVVRSSHADMAAPQTLALLKTVTIVLG
VFIVCWLPAFSILLLDYACPVHSCPILYKAHYFFAVSTLNSLLNPVIYTWRSRDLRREVL
RPLQCWRPGVGVQGRRRGGTPGHHLLPLRSSSSLERGMHMPTSPTFLEGNTVV

BDBM41668

n/a

Name

BDBM41668

Synonyms:

1-(3-imidazol-1-ylpropyl)-2-imino-10-methyl-5-oxo-N-(2-phenylethyl)dipyrido[3,4-c:1',2'-f]pyrimidine-3-carboxamide | 1-(3-imidazol-1-ylpropyl)-2-imino-5-keto-10-methyl-N-phenethyl-dipyrido[3,4-c:1',2'-f]pyrimidine-3-carboxamide | 1-[3-(1-imidazolyl)propyl]-2-imino-10-methyl-5-oxo-N-(2-phenylethyl)-3-dipyrido[3,4-c:1',2'-f]pyrimidinecarboxamide | 2-azanylidene-1-(3-imidazol-1-ylpropyl)-10-methyl-5-oxidanylidene-N-(2-phenylethyl)dipyrido[3,4-c:1',2'-f]pyrimidine-3-carboxamide | MLS000519295 | SMR000129714 | cid_5201463

Type

Small organic molecule

Emp. Form.

C27H27N7O2

Mol. Mass.

481.549

SMILES

Cc1cccn2c1nc1n(CCCn3ccnc3)c(=N)c(cc1c2=O)C(=O)NCCc1ccccc1

Structure