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Reaction Details
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TargetSphingosine 1-phosphate receptor 2
LigandBDBM41710
Substrate/Competitorn/a
Meas. Tech.Dose Response Cell Based Assay for Agonists of the S1P2 Receptor of Purchased Analogues
EC50>30000±n/a nM
Citation PubChem, PC Dose Response Cell Based Assay for Agonists of the S1P2 Receptor of Purchased Analogues PubChem Bioassay(2007)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Sphingosine 1-phosphate receptor 2
Name:Sphingosine 1-phosphate receptor 2
Synonyms:EDG5 | S1P2 | S1PR2 | S1PR2_HUMAN | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor Edg-5 | Sphingosine-1-phosphate receptor 2 | ndothelial differentiation G-protein coupled receptor 5
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:38883.16
Organism:Homo sapiens (Human)
Description:Membranes isolated from S1P2-transfected CHO cells were used in ligand binding assay.
Residue:353
Sequence:
MGSLYSEYLNPNKVQEHYNYTKETLETQETTSRQVASAFIVILCCAIVVENLLVLIAVAR
NSKFHSAMYLFLGNLAASDLLAGVAFVANTLLSGSVTLRLTPVQWFAREGSAFITLSASV
FSLLAIAIERHVAIAKVKLYGSDKSCRMLLLIGASWLISLVLGGLPILGWNCLGHLEACS
TVLPLYAKHYVLCVVTIFSIILLAIVALYVRIYCVVRSSHADMAAPQTLALLKTVTIVLG
VFIVCWLPAFSILLLDYACPVHSCPILYKAHYFFAVSTLNSLLNPVIYTWRSRDLRREVL
RPLQCWRPGVGVQGRRRGGTPGHHLLPLRSSSSLERGMHMPTSPTFLEGNTVV
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  Blast E-value cutoff:
BDBM41710
n/a
NameBDBM41710
Synonyms:2-[[2-(1-benzyl-2,5-dimethyl-pyrrol-3-yl)-2-keto-ethyl]-methyl-amino]-N-cyclopropyl-acetamide | 2-[[2-(1-benzyl-2,5-dimethylpyrrol-3-yl)-2-oxoethyl]-methylamino]-N-cyclopropylacetamide | N-cyclopropyl-2-[[2-[2,5-dimethyl-1-(phenylmethyl)-3-pyrrolyl]-2-oxoethyl]-methylamino]acetamide | N-cyclopropyl-2-[[2-[2,5-dimethyl-1-(phenylmethyl)pyrrol-3-yl]-2-oxidanylidene-ethyl]-methyl-amino]ethanamide | SR-01000759106-1 | cid_8909761
TypeSmall organic molecule
Emp. Form.C21H27N3O2
Mol. Mass.353.458
SMILESCN(CC(=O)NC1CC1)CC(=O)c1cc(C)n(Cc2ccccc2)c1C
Structure
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