Reaction Details |
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Target | Sphingosine 1-phosphate receptor 2 |
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Ligand | BDBM41719 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose Response Cell Based Assay for Agonists of the S1P2 Receptor of Purchased Analogues |
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EC50 | >30000±n/a nM |
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Citation | PubChem, PC Dose Response Cell Based Assay for Agonists of the S1P2 Receptor of Purchased Analogues PubChem Bioassay(2007)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Sphingosine 1-phosphate receptor 2 |
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Name: | Sphingosine 1-phosphate receptor 2 |
Synonyms: | EDG5 | S1P2 | S1PR2 | S1PR2_HUMAN | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor Edg-5 | Sphingosine-1-phosphate receptor 2 | ndothelial differentiation G-protein coupled receptor 5 |
Type: | G Protein-Coupled Receptor (GPCR) |
Mol. Mass.: | 38883.16 |
Organism: | Homo sapiens (Human) |
Description: | Membranes isolated from S1P2-transfected CHO cells were used in ligand binding assay. |
Residue: | 353 |
Sequence: | MGSLYSEYLNPNKVQEHYNYTKETLETQETTSRQVASAFIVILCCAIVVENLLVLIAVAR
NSKFHSAMYLFLGNLAASDLLAGVAFVANTLLSGSVTLRLTPVQWFAREGSAFITLSASV
FSLLAIAIERHVAIAKVKLYGSDKSCRMLLLIGASWLISLVLGGLPILGWNCLGHLEACS
TVLPLYAKHYVLCVVTIFSIILLAIVALYVRIYCVVRSSHADMAAPQTLALLKTVTIVLG
VFIVCWLPAFSILLLDYACPVHSCPILYKAHYFFAVSTLNSLLNPVIYTWRSRDLRREVL
RPLQCWRPGVGVQGRRRGGTPGHHLLPLRSSSSLERGMHMPTSPTFLEGNTVV
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BDBM41719 |
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n/a |
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Name | BDBM41719 |
Synonyms: | 1-[2,5-dimethyl-1-(phenylmethyl)pyrrol-3-yl]-2-(4-ethanoylphenoxy)ethanone | 2-(4-acetylphenoxy)-1-(1-benzyl-2,5-dimethyl-pyrrol-3-yl)ethanone | 2-(4-acetylphenoxy)-1-(1-benzyl-2,5-dimethylpyrrol-3-yl)ethanone | 2-(4-acetylphenoxy)-1-[2,5-dimethyl-1-(phenylmethyl)-3-pyrrolyl]ethanone | SR-01000759118-1 | cid_7763884 |
Type | Small organic molecule |
Emp. Form. | C23H23NO3 |
Mol. Mass. | 361.4336 |
SMILES | CC(=O)c1ccc(OCC(=O)c2cc(C)n(Cc3ccccc3)c2C)cc1 |
Structure |
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