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TargetBcl-2-related protein A1
LigandBDBM39118
Substrate/Competitorn/a
Meas. Tech.In Vitro Bfl-1 Dose Response Fluorescence Polarization Assay for SAR Study
IC50 6780±1900 nM
Citation PubChem, PC In Vitro Bfl-1 Dose Response Fluorescence Polarization Assay for SAR Study PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Bcl-2-related protein A1
Name:Bcl-2-related protein A1
Synonyms:A1 | A1-A | B-cell leukemia/lymphoma 2 related protein A1a | B2LA1_MOUSE | Bcl2a1 | Bcl2a1a | Bfl-1 | Bfl1 | Hemopoietic-specific early response protein | Protein BFL-1
Type:Apoptosis regulator protein
Mol. Mass.:19909.74
Organism:Mus musculus (Mouse)
Description:gi_11024684
Residue:172
Sequence:
MAESELMHIHSLAEHYLQYVLQVPAFESAPSQACRVLQRVAFSVQKEVEKNLKSYLDDFH
VESIDTARIIFNQVMEKEFEDGIINWGRIVTIFAFGGVLLKKLPQEQIALDVCAYKQVSS
FVAEFIMNNTGEWIRQNGGWEDGFIKKFEPKSGWLTFLQMTGQIWEMLFLLK
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BDBM39118
n/a
NameBDBM39118
Synonyms:2-mesyl-4-(3-methoxyphenyl)-6-(trifluoromethyl)pyrimidine | 4-(3-methoxyphenyl)-2-methylsulfonyl-6-(trifluoromethyl)pyrimidine | MLS-0066988.0001 | US11725000, Compound 52 | cid_751044
TypeSmall organic molecule
Emp. Form.C13H11F3N2O3S
Mol. Mass.332.298
SMILESCOc1cccc(c1)-c1cc(nc(n1)S(C)(=O)=O)C(F)(F)F
Structure
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