Reaction Details | |||
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Target | Bcl-2-related protein A1 | ||
Ligand | BDBM34180 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | In Vitro Bfl-1 Dose Response Fluorescence Polarization Assay for SAR Study | ||
IC50 | 5390±820 nM | ||
Citation | PubChem, PC In Vitro Bfl-1 Dose Response Fluorescence Polarization Assay for SAR Study PubChem Bioassay(2008)[AID] | ||
More Info.: | Get all data from this article, Solution Info, Assay Method | ||
Bcl-2-related protein A1 | |||
Name: | Bcl-2-related protein A1 | ||
Synonyms: | A1 | A1-A | B-cell leukemia/lymphoma 2 related protein A1a | B2LA1_MOUSE | Bcl2a1 | Bcl2a1a | Bfl-1 | Bfl1 | Hemopoietic-specific early response protein | Protein BFL-1 | ||
Type: | Apoptosis regulator protein | ||
Mol. Mass.: | 19909.74 | ||
Organism: | Mus musculus (Mouse) | ||
Description: | gi_11024684 | ||
Residue: | 172 | ||
Sequence: |
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BDBM34180 | |||
n/a | |||
Name | BDBM34180 | ||
Synonyms: | 3-(3,4-dimethoxyphenyl)-1-[(pentafluorophenyl)sulfonyl]-1H-pyrazol-5-amine | 5-(3,4-dimethoxyphenyl)-2-(2,3,4,5,6-pentafluorophenyl)sulfonyl-3-pyrazolamine | 5-(3,4-dimethoxyphenyl)-2-(2,3,4,5,6-pentafluorophenyl)sulfonylpyrazol-3-amine | 5-(3,4-dimethoxyphenyl)-2-[2,3,4,5,6-pentakis(fluoranyl)phenyl]sulfonyl-pyrazol-3-amine | MLS000045819 | SMR000028216 | [5-(3,4-dimethoxyphenyl)-2-(2,3,4,5,6-pentafluorophenyl)sulfonyl-pyrazol-3-yl]amine | cid_3237441 | ||
Type | Small organic molecule | ||
Emp. Form. | C17H12F5N3O4S | ||
Mol. Mass. | 449.352 | ||
SMILES | COc1ccc(cc1OC)-c1cc(N)n(n1)S(=O)(=O)c1c(F)c(F)c(F)c(F)c1F | ||
Structure |