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TargetBcl-2-related protein A1
LigandBDBM39173
Substrate/Competitorn/a
Meas. Tech.In Vitro Bfl-1 Dose Response Fluorescence Polarization Assay for SAR Study
IC50 4680±950 nM
Citation PubChem, PC In Vitro Bfl-1 Dose Response Fluorescence Polarization Assay for SAR Study PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Bcl-2-related protein A1
Name:Bcl-2-related protein A1
Synonyms:A1 | A1-A | B-cell leukemia/lymphoma 2 related protein A1a | B2LA1_MOUSE | Bcl2a1 | Bcl2a1a | Bfl-1 | Bfl1 | Hemopoietic-specific early response protein | Protein BFL-1
Type:Apoptosis regulator protein
Mol. Mass.:19909.74
Organism:Mus musculus (Mouse)
Description:gi_11024684
Residue:172
Sequence:
MAESELMHIHSLAEHYLQYVLQVPAFESAPSQACRVLQRVAFSVQKEVEKNLKSYLDDFH
VESIDTARIIFNQVMEKEFEDGIINWGRIVTIFAFGGVLLKKLPQEQIALDVCAYKQVSS
FVAEFIMNNTGEWIRQNGGWEDGFIKKFEPKSGWLTFLQMTGQIWEMLFLLK
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BDBM39173
n/a
NameBDBM39173
Synonyms:3-[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-4-chloro-1-(4-nitrophenyl)pyrrole-2,5-dione | 3-[4-(1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-4-chloranyl-1-(4-nitrophenyl)pyrrole-2,5-dione | 3-[4-(1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-4-chloro-1-(4-nitrophenyl)pyrrole-2,5-dione | 3-chloro-1-(4-nitrophenyl)-4-(4-piperonylpiperazino)-3-pyrroline-2,5-quinone | MLS-0111727.0001 | cid_16654756
TypeSmall organic molecule
Emp. Form.C22H19ClN4O6
Mol. Mass.470.862
SMILES[O-][N+](=O)c1ccc(cc1)N1C(=O)C(Cl)=C(N2CCN(Cc3ccc4OCOc4c3)CC2)C1=O |t:14|
Structure
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