| Reaction Details |
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 | Report a problem with these data |
| Target | Galanin receptor type 2 |
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| Ligand | BDBM42058 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2) |
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| IC50 | >42000±n/a nM |
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| Citation |  PubChem, PC Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2) PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Galanin receptor type 2 |
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| Name: | Galanin receptor type 2 |
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| Synonyms: | GALNR2 | GALR2 | GALR2_HUMAN | Galanin R2 | Galanin receptor 2 | Galanin receptor type 2 | Galanin receptor type 2 (GAL2-R) (GALR2). |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 41724.40 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Galanin R2 GALR2 HUMAN::O43603 |
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| Residue: | 387 |
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| Sequence: | MNVSGCPGAGNASQAGGGGGWHPEAVIVPLLFALIFLVGTVGNTLVLAVLLRGGQAVSTT
NLFILNLGVADLCFILCCVPFQATIYTLDGWVFGSLLCKAVHFLIFLTMHASSFTLAAVS
LDRYLAIRYPLHSRELRTPRNALAAIGLIWGLSLLFSGPYLSYYRQSQLANLTVCHPAWS
APRRRAMDICTFVFSYLLPVLVLGLTYARTLRYLWRAVDPVAAGSGARRAKRKVTRMILI
VAALFCLCWMPHHALILCVWFGQFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFR
KGFRTICAGLLGRAPGRASGRVCAAARGTHSGSVLERESSDLLHMSEAAGALRPCPGASQ
PCILEPCPGPSWQGPKAGDSILTVDVA
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| BDBM42058 |
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| n/a |
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| Name | BDBM42058 |
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| Synonyms: | (2-Cyclohex-1-enyl-ethyl)-(5H-pyrimido[5,4-b]indol-4-yl)-amine | 2-(cyclohexen-1-yl)ethyl-(5H-pyrimid[5,4-b]indol-4-yl)amine | MLS000580267 | N-[2-(1-cyclohexenyl)ethyl]-5H-pyrimido[5,4-b]indol-4-amine | N-[2-(cyclohexen-1-yl)ethyl]-5H-pyrimido[5,4-b]indol-4-amine | SMR000220470 | cid_944164 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H20N4 |
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| Mol. Mass. | 292.3782 |
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| SMILES | C(CC1=CCCCC1)Nc1ncnc2c3ccccc3[nH]c12 |t:2| |
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| Structure | 
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