| Reaction Details |
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 | Report a problem with these data |
| Target | Galanin receptor type 2 |
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| Ligand | BDBM42037 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity |
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| IC50 | >42000±n/a nM |
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| Citation |  PubChem, PC Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Galanin receptor type 2 |
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| Name: | Galanin receptor type 2 |
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| Synonyms: | GALNR2 | GALR2 | GALR2_HUMAN | Galanin R2 | Galanin receptor 2 | Galanin receptor type 2 | Galanin receptor type 2 (GAL2-R) (GALR2). |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 41724.40 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Galanin R2 GALR2 HUMAN::O43603 |
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| Residue: | 387 |
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| Sequence: | MNVSGCPGAGNASQAGGGGGWHPEAVIVPLLFALIFLVGTVGNTLVLAVLLRGGQAVSTT
NLFILNLGVADLCFILCCVPFQATIYTLDGWVFGSLLCKAVHFLIFLTMHASSFTLAAVS
LDRYLAIRYPLHSRELRTPRNALAAIGLIWGLSLLFSGPYLSYYRQSQLANLTVCHPAWS
APRRRAMDICTFVFSYLLPVLVLGLTYARTLRYLWRAVDPVAAGSGARRAKRKVTRMILI
VAALFCLCWMPHHALILCVWFGQFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFR
KGFRTICAGLLGRAPGRASGRVCAAARGTHSGSVLERESSDLLHMSEAAGALRPCPGASQ
PCILEPCPGPSWQGPKAGDSILTVDVA
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| BDBM42037 |
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| n/a |
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| Name | BDBM42037 |
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| Synonyms: | 4-(1-piperidinyl)-5H-pyrimido[5,4-b]indole | 4-piperidin-1-yl-5H-pyrimido[5,4-b]indole | 4-piperidino-5H-pyrimid[5,4-b]indole | MLS000027106 | SMR000008850 | cid_646579 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H16N4 |
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| Mol. Mass. | 252.3143 |
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| SMILES | C1CCN(CC1)c1ncnc2c3ccccc3[nH]c12 |
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| Structure | 
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