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TargetGalanin receptor type 2
LigandBDBM42069
Substrate/Competitorn/a
Meas. Tech.Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity
IC50 7528±n/a nM
Citation PubChem, PC Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Galanin receptor type 2
Name:Galanin receptor type 2
Synonyms:GALNR2 | GALR2 | GALR2_HUMAN | Galanin R2 | Galanin receptor 2 | Galanin receptor type 2 | Galanin receptor type 2 (GAL2-R) (GALR2).
Type:Enzyme Catalytic Domain
Mol. Mass.:41724.40
Organism:Homo sapiens (Human)
Description:Galanin R2 GALR2 HUMAN::O43603
Residue:387
Sequence:
MNVSGCPGAGNASQAGGGGGWHPEAVIVPLLFALIFLVGTVGNTLVLAVLLRGGQAVSTT
NLFILNLGVADLCFILCCVPFQATIYTLDGWVFGSLLCKAVHFLIFLTMHASSFTLAAVS
LDRYLAIRYPLHSRELRTPRNALAAIGLIWGLSLLFSGPYLSYYRQSQLANLTVCHPAWS
APRRRAMDICTFVFSYLLPVLVLGLTYARTLRYLWRAVDPVAAGSGARRAKRKVTRMILI
VAALFCLCWMPHHALILCVWFGQFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFR
KGFRTICAGLLGRAPGRASGRVCAAARGTHSGSVLERESSDLLHMSEAAGALRPCPGASQ
PCILEPCPGPSWQGPKAGDSILTVDVA
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  Blast E-value cutoff:
BDBM42069
n/a
NameBDBM42069
Synonyms:2-acetamido-4,5-dinitro-benzoic acid ethyl ester | 2-acetamido-4,5-dinitrobenzoic acid ethyl ester | MLS000698400 | SMR000224624 | cid_4104905 | ethyl 2-(acetylamino)-4,5-dinitrobenzoate | ethyl 2-acetamido-4,5-dinitro-benzoate | ethyl 2-acetamido-4,5-dinitrobenzoate
TypeSmall organic molecule
Emp. Form.C11H11N3O7
Mol. Mass.297.2209
SMILESCCOC(=O)c1cc(c(cc1NC(C)=O)[N+]([O-])=O)[N+]([O-])=O
Structure
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