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TargetNeuropeptide Y receptor type 2
LigandBDBM38831
Substrate/Competitorn/a
Meas. Tech.Dose response counterscreen assay for neuropeptide Y receptor Y1 (NPY-Y1): Cell-based high throughput assay to measure NPY-Y2 antagonism
IC50>35000±n/a nM
Citation PubChem, PC Dose response counterscreen assay for neuropeptide Y receptor Y1 (NPY-Y1): Cell-based high throughput assay to measure NPY-Y2 antagonism PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Neuropeptide Y receptor type 2
Name:Neuropeptide Y receptor type 2
Synonyms:NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2
Type:Enzyme Catalytic Domain
Mol. Mass.:42734.65
Organism:Homo sapiens (Human)
Description:NPY-Y2 NPY2R HUMAN::P49146
Residue:381
Sequence:
MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSI
ILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAK
KNLEVRKNSGPNDSFTEATNV
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BDBM38831
n/a
NameBDBM38831
Synonyms:3-methyl-1-phenyl-1H-thieno[2,3-c]pyrazole-5-carboxylic acid | 3-methyl-1-phenyl-5-thieno[2,3-c]pyrazolecarboxylic acid | 3-methyl-1-phenyl-thieno[2,3-c]pyrazole-5-carboxylic acid | 3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carboxylic acid | MLS000099719 | SMR000071493 | cid_802154
TypeSmall organic molecule
Emp. Form.C13H10N2O2S
Mol. Mass.258.296
SMILESCc1nn(-c2ccccc2)c2sc(cc12)C(O)=O
Structure
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