| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Neuropeptide Y receptor type 2 |
|---|
| Ligand | BDBM42418 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Dose response counterscreen assay for neuropeptide Y receptor Y1 (NPY-Y1): Cell-based high throughput assay to measure NPY-Y2 antagonism |
|---|
| IC50 | >35000±n/a nM |
|---|
| Citation |  PubChem, PC Dose response counterscreen assay for neuropeptide Y receptor Y1 (NPY-Y1): Cell-based high throughput assay to measure NPY-Y2 antagonism PubChem Bioassay(2008)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Neuropeptide Y receptor type 2 |
|---|
| Name: | Neuropeptide Y receptor type 2 |
|---|
| Synonyms: | NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 42734.65 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | NPY-Y2 NPY2R HUMAN::P49146 |
|---|
| Residue: | 381 |
|---|
| Sequence: | MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSI
ILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAK
KNLEVRKNSGPNDSFTEATNV
|
|
|
|---|
| BDBM42418 |
|---|
| n/a |
|---|
| Name | BDBM42418 |
|---|
| Synonyms: | 1-(1-tert-butyl-1,2,3,4-tetrazol-5-yl)-N-(furan-2-ylmethyl)-N-(phenylmethyl)-1-[4-(trifluoromethyl)phenyl]methanamine | 1-(1-tert-butyl-5-tetrazolyl)-N-(2-furanylmethyl)-N-(phenylmethyl)-1-[4-(trifluoromethyl)phenyl]methanamine | Benzyl-[(1-tert-butyl-1H-tetrazol-5-yl)-(4-trifluoromethyl-phenyl)-methyl]-furan-2-ylmethyl-amine | MLS000528002 | N-benzyl-1-(1-tert-butyltetrazol-5-yl)-N-(furan-2-ylmethyl)-1-[4-(trifluoromethyl)phenyl]methanamine | SMR000120576 | benzyl-[(1-tert-butyltetrazol-5-yl)-[4-(trifluoromethyl)phenyl]methyl]-(2-furfuryl)amine | cid_3229320 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C25H26F3N5O |
|---|
| Mol. Mass. | 469.502 |
|---|
| SMILES | CC(C)(C)n1nnnc1C(N(Cc1ccco1)Cc1ccccc1)c1ccc(cc1)C(F)(F)F |
|---|
| Structure | 
|
|---|
Search and Browse
