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TargetNeuropeptide Y receptor type 2
LigandBDBM42435
Substrate/Competitorn/a
Meas. Tech.Dose response counterscreen assay for neuropeptide Y receptor Y1 (NPY-Y1): Cell-based high throughput assay to measure NPY-Y2 antagonism
IC50 10590±n/a nM
Citation PubChem, PC Dose response counterscreen assay for neuropeptide Y receptor Y1 (NPY-Y1): Cell-based high throughput assay to measure NPY-Y2 antagonism PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Neuropeptide Y receptor type 2
Name:Neuropeptide Y receptor type 2
Synonyms:NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2
Type:Enzyme Catalytic Domain
Mol. Mass.:42734.65
Organism:Homo sapiens (Human)
Description:NPY-Y2 NPY2R HUMAN::P49146
Residue:381
Sequence:
MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSI
ILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAK
KNLEVRKNSGPNDSFTEATNV
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BDBM42435
n/a
NameBDBM42435
Synonyms:(4-methylphenyl)methyl 5-amino-2-phenyltriazole-4-carboxylate | (4-methylphenyl)methyl 5-azanyl-2-phenyl-1,2,3-triazole-4-carboxylate | 4-methylbenzyl 5-amino-2-phenyl-2H-1,2,3-triazole-4-carboxylate | 5-amino-2-phenyl-4-triazolecarboxylic acid (4-methylphenyl)methyl ester | 5-amino-2-phenyl-triazole-4-carboxylic acid (4-methylbenzyl) ester | MLS000729082 | SMR000307360 | cid_1504749
TypeSmall organic molecule
Emp. Form.C17H16N4O2
Mol. Mass.308.3345
SMILESCc1ccc(COC(=O)c2nn(nc2N)-c2ccccc2)cc1
Structure
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