| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide Y receptor type 2 |
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| Ligand | BDBM42437 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response counterscreen assay for neuropeptide Y receptor Y1 (NPY-Y1): Cell-based high throughput assay to measure NPY-Y2 antagonism |
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| IC50 | >35000±n/a nM |
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| Citation |  PubChem, PC Dose response counterscreen assay for neuropeptide Y receptor Y1 (NPY-Y1): Cell-based high throughput assay to measure NPY-Y2 antagonism PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Neuropeptide Y receptor type 2 |
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| Name: | Neuropeptide Y receptor type 2 |
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| Synonyms: | NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 42734.65 |
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| Organism: | Homo sapiens (Human) |
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| Description: | NPY-Y2 NPY2R HUMAN::P49146 |
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| Residue: | 381 |
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| Sequence: | MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSI
ILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAK
KNLEVRKNSGPNDSFTEATNV
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| BDBM42437 |
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| n/a |
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| Name | BDBM42437 |
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| Synonyms: | 1-[1-acetyl-5-(4-chlorophenyl)-6-(4-methoxyphenyl)-2-methyl-1,2,5,6-tetrahydro-1,2,4,5-tetrazin-3-yl]ethanone | 1-[2-acetyl-4-(4-chlorophenyl)-3-(4-methoxyphenyl)-1-methyl-3H-1,2,4,5-tetrazin-6-yl]ethanone | 1-[4-(4-chlorophenyl)-2-ethanoyl-3-(4-methoxyphenyl)-1-methyl-3H-1,2,4,5-tetrazin-6-yl]ethanone | MLS000727503 | SMR000306200 | cid_539575 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H21ClN4O3 |
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| Mol. Mass. | 400.859 |
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| SMILES | COc1ccc(cc1)C1N(N=C(N(C)N1C(C)=O)C(C)=O)c1ccc(Cl)cc1 |c:11| |
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| Structure | 
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