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TargetCell division control protein 42 homolog
LigandBDBM43207
Substrate/Competitorn/a
Meas. Tech.Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant
EC50 5854±n/a nM
Citation PubChem, PC Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Cell division control protein 42 homolog
Name:Cell division control protein 42 homolog
Synonyms:CDC42 | CDC42_HUMAN | Cell division control protein 42 homolog | G25K GTP-binding protein | cell division cycle 42 (GTP binding protein, 25kDa)
Type:PROTEIN
Mol. Mass.:21258.36
Organism:Homo sapiens (Human)
Description:ChEMBL_652970
Residue:191
Sequence:
MQTIKCVVVGDGAVGKTCLLISYTTNKFPSEYVPTVFDNYAVTVMIGGEPYTLGLFDTAG
QEDYDRLRPLSYPQTDVFLVCFSVVSPSSFENVKEKWVPEITHHCPKTPFLLVGTQIDLR
DDPSTIEKLAKNKQKPITPETAEKLARDLKAVKYVECSALTQKGLKNVFDEAILAALEPP
EPKKSRRCVLL
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BDBM43207
n/a
NameBDBM43207
Synonyms:2-[(2,6-dichlorobenzyl)amino]-3-methyl-butyric acid | 2-[(2,6-dichlorophenyl)methylamino]-3-methylbutanoic acid | 2-[[2,6-bis(chloranyl)phenyl]methylamino]-3-methyl-butanoic acid | MLS000095936 | N-(2,6-dichlorobenzyl)valine | SMR000031484 | cid_3237092
TypeSmall organic molecule
Emp. Form.C12H15Cl2NO2
Mol. Mass.276.159
SMILESCC(C)C(NCc1c(Cl)cccc1Cl)C(O)=O
Structure
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