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TargetSignal transducer and activator of transcription 3 [702-738,740-752]
LigandBDBM43021
Substrate/Competitorn/a
Meas. Tech.Dose response cell-based assay to measure STAT3 activation
IC50>18560±n/a nM
Citation PubChem, PC Dose response cell-based assay to measure STAT3 activation PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Signal transducer and activator of transcription 3 [702-738,740-752]
Name:Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:APRF | STAT3 | STAT3_HUMAN
Type:Enzyme Catalytic Domain
Mol. Mass.:5263.93
Organism:Homo sapiens (Human)
Description:gi_13272532
Residue:50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
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BDBM43021
n/a
NameBDBM43021
Synonyms:3-[(5-bromothiophene-2-carbonyl)amino]thiophene-2-carboxylic acid methyl ester | 3-[[(5-bromo-2-thiophenyl)-oxomethyl]amino]-2-thiophenecarboxylic acid methyl ester | MLS000538431 | SMR000144468 | cid_1246013 | methyl 3-[(5-bromanylthiophen-2-yl)carbonylamino]thiophene-2-carboxylate | methyl 3-[(5-bromothiophene-2-carbonyl)amino]thiophene-2-carboxylate | methyl 3-{[(5-bromo-2-thienyl)carbonyl]amino}-2-thiophenecarboxylate
TypeSmall organic molecule
Emp. Form.C11H8BrNO3S2
Mol. Mass.346.22
SMILESCOC(=O)c1sccc1NC(=O)c1ccc(Br)s1
Structure
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