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TargetSignal transducer and activator of transcription 3 [702-738,740-752]
LigandBDBM43661
Substrate/Competitorn/a
Meas. Tech.Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation
EC50>55700±n/a nM
Citation PubChem, PC Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Signal transducer and activator of transcription 3 [702-738,740-752]
Name:Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:APRF | STAT3 | STAT3_HUMAN
Type:Enzyme Catalytic Domain
Mol. Mass.:5263.93
Organism:Homo sapiens (Human)
Description:gi_13272532
Residue:50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
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BDBM43661
n/a
NameBDBM43661
Synonyms:4-Methyl-thiazole-5-carboxylic acid (4,5,6,7-tetrahydro-benzothiazol-2-yl)-amide | 4-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1,3-thiazole-5-carboxamide | 4-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-5-thiazolecarboxamide | 4-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)thiazole-5-carboxamide | MLS000074500 | SMR000007300 | cid_653744
TypeSmall organic molecule
Emp. Form.C12H13N3OS2
Mol. Mass.279.381
SMILESCc1ncsc1C(=O)Nc1nc2CCCCc2s1
Structure
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