| Reaction Details |
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 | Report a problem with these data |
| Target | Sphingosine 1-phosphate receptor 2 |
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| Ligand | BDBM41680 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Counter screen for S1P2 Agonists: Dose Response High Throughput Cell-Based Screen to Identify Activators of CRE-BLA |
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| EC50 | 3349±n/a nM |
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| Citation |  PubChem, PC Counter screen for S1P2 Agonists: Dose Response High Throughput Cell-Based Screen to Identify Activators of CRE-BLA PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Sphingosine 1-phosphate receptor 2 |
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| Name: | Sphingosine 1-phosphate receptor 2 |
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| Synonyms: | EDG5 | S1P2 | S1PR2 | S1PR2_HUMAN | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor Edg-5 | Sphingosine-1-phosphate receptor 2 | ndothelial differentiation G-protein coupled receptor 5 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 38883.16 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Membranes isolated from S1P2-transfected CHO cells were used in ligand binding assay. |
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| Residue: | 353 |
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| Sequence: | MGSLYSEYLNPNKVQEHYNYTKETLETQETTSRQVASAFIVILCCAIVVENLLVLIAVAR
NSKFHSAMYLFLGNLAASDLLAGVAFVANTLLSGSVTLRLTPVQWFAREGSAFITLSASV
FSLLAIAIERHVAIAKVKLYGSDKSCRMLLLIGASWLISLVLGGLPILGWNCLGHLEACS
TVLPLYAKHYVLCVVTIFSIILLAIVALYVRIYCVVRSSHADMAAPQTLALLKTVTIVLG
VFIVCWLPAFSILLLDYACPVHSCPILYKAHYFFAVSTLNSLLNPVIYTWRSRDLRREVL
RPLQCWRPGVGVQGRRRGGTPGHHLLPLRSSSSLERGMHMPTSPTFLEGNTVV
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| BDBM41680 |
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| n/a |
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| Name | BDBM41680 |
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| Synonyms: | 1-(4-Chloro-phenyl)-5-furan-2-yl-3-thiophen-2-yl-4,5-dihydro-1H-pyrazole | 1-(4-chlorophenyl)-5-(2-furyl)-3-(2-thienyl)-2-pyrazoline | 2-(4-chlorophenyl)-3-(2-furanyl)-5-thiophen-2-yl-3,4-dihydropyrazole | 2-(4-chlorophenyl)-3-(furan-2-yl)-5-thiophen-2-yl-3,4-dihydropyrazole | MLS000566481 | SMR000174942 | cid_2842931 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H13ClN2OS |
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| Mol. Mass. | 328.816 |
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| SMILES | Clc1ccc(cc1)N1N=C(CC1c1ccco1)c1cccs1 |c:9| |
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| Structure | 
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