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TargetGlutathione S-transferase Mu 1
LigandBDBM46294
Substrate/Competitorn/a
Meas. Tech.Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer)
EC50 27980±n/a nM
Citation PubChem, PC Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer) PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Glutathione S-transferase Mu 1
Name:Glutathione S-transferase Mu 1
Synonyms:GST class-mu 1 | GST1 | GSTM1 | GSTM1-1 | GSTM1_HUMAN | GSTM1a-1a | GSTM1b-1b | GTH4 | Glutathione S-transferase Mu 1 | HB subunit 4 | glutathione S-transferase
Type:PROTEIN
Mol. Mass.:25712.03
Organism:Homo sapiens (Human)
Description:ChEMBL_799596
Residue:218
Sequence:
MPMILGYWDIRGLAHAIRLLLEYTDSSYEEKKYTMGDAPDYDRSQWLNEKFKLGLDFPNL
PYLIDGAHKITQSNAILCYIARKHNLCGETEEEKIRVDILENQTMDNHMQLGMICYNPEF
EKLKPKYLEELPEKLKLYSEFLGKRPWFAGNKITFVDFLVYDVLDLHRIFEPKCLDAFPN
LKDFISRFEGLEKISAYMKSSRFLPRPVFSKMAVWGNK
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BDBM46294
n/a
NameBDBM46294
Synonyms:4-keto-5-methyl-3H-thieno[2,3-d]pyrimidine-6-carboxylic acid methyl ester | 5-Methyl-4-oxo-3,4-dihydro-thieno[2,3-d]pyrimidine-6-carboxylic acid methyl ester | 5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylic acid methyl ester | MLS000067670 | SMR000125022 | cid_725279 | methyl 5-methyl-4-oxidanylidene-3H-thieno[2,3-d]pyrimidine-6-carboxylate | methyl 5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
TypeSmall organic molecule
Emp. Form.C9H8N2O3S
Mol. Mass.224.236
SMILESCOC(=O)c1sc2nc[nH]c(=O)c2c1C
Structure
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