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TargetGlutathione S-transferase Mu 1
LigandBDBM46298
Substrate/Competitorn/a
Meas. Tech.Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer)
EC50 26410±n/a nM
Citation PubChem, PC Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer) PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Glutathione S-transferase Mu 1
Name:Glutathione S-transferase Mu 1
Synonyms:GST class-mu 1 | GST1 | GSTM1 | GSTM1-1 | GSTM1_HUMAN | GSTM1a-1a | GSTM1b-1b | GTH4 | Glutathione S-transferase Mu 1 | HB subunit 4 | glutathione S-transferase
Type:PROTEIN
Mol. Mass.:25712.03
Organism:Homo sapiens (Human)
Description:ChEMBL_799596
Residue:218
Sequence:
MPMILGYWDIRGLAHAIRLLLEYTDSSYEEKKYTMGDAPDYDRSQWLNEKFKLGLDFPNL
PYLIDGAHKITQSNAILCYIARKHNLCGETEEEKIRVDILENQTMDNHMQLGMICYNPEF
EKLKPKYLEELPEKLKLYSEFLGKRPWFAGNKITFVDFLVYDVLDLHRIFEPKCLDAFPN
LKDFISRFEGLEKISAYMKSSRFLPRPVFSKMAVWGNK
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BDBM46298
n/a
NameBDBM46298
Synonyms:2-[(1,1-diketo-1,2-benzothiazol-3-yl)-[(3-methylbenzylidene)amino]amino]ethanol | 2-[(1,1-dioxo-1,2-benzothiazol-3-yl)-[(3-methylphenyl)methylideneamino]amino]ethanol | 2-[[1,1-bis(oxidanylidene)-1,2-benzothiazol-3-yl]-[(3-methylphenyl)methylideneamino]amino]ethanol | 3-methylbenzaldehyde (1,1-dioxido-1,2-benzisothiazol-3-yl)(2-hydroxyethyl)hydrazone | MLS000686259 | SMR000313102 | cid_4421869
TypeSmall organic molecule
Emp. Form.C17H17N3O3S
Mol. Mass.343.4
SMILESCc1cccc(C=NN(CCO)C2=NS(=O)(=O)c3ccccc23)c1 |w:7.7,t:12|
Structure
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