Reaction Details |
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Target | Glutathione S-transferase Mu 1 |
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Ligand | BDBM32330 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer) |
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EC50 | 4780±n/a nM |
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Citation | PubChem, PC Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer) PubChem Bioassay(2008)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Glutathione S-transferase Mu 1 |
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Name: | Glutathione S-transferase Mu 1 |
Synonyms: | GST class-mu 1 | GST1 | GSTM1 | GSTM1-1 | GSTM1_HUMAN | GSTM1a-1a | GSTM1b-1b | GTH4 | Glutathione S-transferase Mu 1 | HB subunit 4 | glutathione S-transferase |
Type: | PROTEIN |
Mol. Mass.: | 25712.03 |
Organism: | Homo sapiens (Human) |
Description: | ChEMBL_799596 |
Residue: | 218 |
Sequence: | MPMILGYWDIRGLAHAIRLLLEYTDSSYEEKKYTMGDAPDYDRSQWLNEKFKLGLDFPNL
PYLIDGAHKITQSNAILCYIARKHNLCGETEEEKIRVDILENQTMDNHMQLGMICYNPEF
EKLKPKYLEELPEKLKLYSEFLGKRPWFAGNKITFVDFLVYDVLDLHRIFEPKCLDAFPN
LKDFISRFEGLEKISAYMKSSRFLPRPVFSKMAVWGNK
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BDBM32330 |
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n/a |
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Name | BDBM32330 |
Synonyms: | (2Z)-2-(5-fluoranyl-2-oxidanylidene-indol-3-yl)-2-(4-methyl-3H-1,3-thiazol-2-ylidene)ethanenitrile | (2Z)-2-(5-fluoro-2-keto-indol-3-yl)-2-(4-methyl-4-thiazolin-2-ylidene)acetonitrile | (2Z)-2-(5-fluoro-2-oxo-3-indolyl)-2-(4-methyl-3H-thiazol-2-ylidene)acetonitrile | (2Z)-2-(5-fluoro-2-oxoindol-3-yl)-2-(4-methyl-3H-1,3-thiazol-2-ylidene)acetonitrile | MLS001011168 | SMR000353171 | cid_16196155 |
Type | Small organic molecule |
Emp. Form. | C14H8FN3OS |
Mol. Mass. | 285.296 |
SMILES | Cc1csc(n1)C(C#N)=C1C(=O)Nc2ccc(F)cc12 |w:9.20| |
Structure |
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