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TargetGlutathione S-transferase Mu 1
LigandBDBM32330
Substrate/Competitorn/a
Meas. Tech.Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer)
EC50 4780±n/a nM
Citation PubChem, PC Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer) PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Glutathione S-transferase Mu 1
Name:Glutathione S-transferase Mu 1
Synonyms:GST class-mu 1 | GST1 | GSTM1 | GSTM1-1 | GSTM1_HUMAN | GSTM1a-1a | GSTM1b-1b | GTH4 | Glutathione S-transferase Mu 1 | HB subunit 4 | glutathione S-transferase
Type:PROTEIN
Mol. Mass.:25712.03
Organism:Homo sapiens (Human)
Description:ChEMBL_799596
Residue:218
Sequence:
MPMILGYWDIRGLAHAIRLLLEYTDSSYEEKKYTMGDAPDYDRSQWLNEKFKLGLDFPNL
PYLIDGAHKITQSNAILCYIARKHNLCGETEEEKIRVDILENQTMDNHMQLGMICYNPEF
EKLKPKYLEELPEKLKLYSEFLGKRPWFAGNKITFVDFLVYDVLDLHRIFEPKCLDAFPN
LKDFISRFEGLEKISAYMKSSRFLPRPVFSKMAVWGNK
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BDBM32330
n/a
NameBDBM32330
Synonyms:(2Z)-2-(5-fluoranyl-2-oxidanylidene-indol-3-yl)-2-(4-methyl-3H-1,3-thiazol-2-ylidene)ethanenitrile | (2Z)-2-(5-fluoro-2-keto-indol-3-yl)-2-(4-methyl-4-thiazolin-2-ylidene)acetonitrile | (2Z)-2-(5-fluoro-2-oxo-3-indolyl)-2-(4-methyl-3H-thiazol-2-ylidene)acetonitrile | (2Z)-2-(5-fluoro-2-oxoindol-3-yl)-2-(4-methyl-3H-1,3-thiazol-2-ylidene)acetonitrile | MLS001011168 | SMR000353171 | cid_16196155
TypeSmall organic molecule
Emp. Form.C14H8FN3OS
Mol. Mass.285.296
SMILESCc1csc(n1)C(C#N)=C1C(=O)Nc2ccc(F)cc12 |w:9.20|
Structure
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