| Reaction Details |
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 | Report a problem with these data |
| Target | Serine/threonine-protein kinase D1 |
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| Ligand | BDBM32360 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Fluorescence polarization assay for PKD inhibitiors-interference assay-57K HTS campaign |
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| IC50 | 16670.80688±n/a nM |
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| Citation |  PubChem, PC Fluorescence polarization assay for PKD inhibitiors-interference assay-57K HTS campaign PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Serine/threonine-protein kinase D1 |
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| Name: | Serine/threonine-protein kinase D1 |
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| Synonyms: | KPCD1_HUMAN | PKD | PKD1 | PRKCM | PRKD1 | Protein kinase C mu | Protein kinase C mu type | Protein kinase C mu type (PRKD1) | Protein kinase C, PKC; classical/novel | Protein kinase D | Protein kinase D (PRKD1) | Serine/threonine-protein kinase D1 (PKD1) | nPKC-D1 | nPKC-mu |
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| Type: | Serine/threonine-protein kinase |
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| Mol. Mass.: | 101705.07 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_115529463 |
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| Residue: | 912 |
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| Sequence: | MSAPPVLRPPSPLLPVAAAAAAAAAALVPGSGPGPAPFLAPVAAPVGGISFHLQIGLSRE
PVLLLQDSSGDYSLAHVREMACSIVDQKFPECGFYGMYDKILLFRHDPTSENILQLVKAA
SDIQEGDLIEVVLSASATFEDFQIRPHALFVHSYRAPAFCDHCGEMLWGLVRQGLKCEGC
GLNYHKRCAFKIPNNCSGVRRRRLSNVSLTGVSTIRTSSAELSTSAPDEPLLQKSPSESF
IGREKRSNSQSYIGRPIHLDKILMSKVKVPHTFVIHSYTRPTVCQYCKKLLKGLFRQGLQ
CKDCRFNCHKRCAPKVPNNCLGEVTINGDLLSPGAESDVVMEEGSDDNDSERNSGLMDDM
EEAMVQDAEMAMAECQNDSGEMQDPDPDHEDANRTISPSTSNNIPLMRVVQSVKHTKRKS
STVMKEGWMVHYTSKDTLRKRHYWRLDSKCITLFQNDTGSRYYKEIPLSEILSLEPVKTS
ALIPNGANPHCFEITTANVVYYVGENVVNPSSPSPNNSVLTSGVGADVARMWEIAIQHAL
MPVIPKGSSVGTGTNLHRDISVSISVSNCQIQENVDISTVYQIFPDEVLGSGQFGIVYGG
KHRKTGRDVAIKIIDKLRFPTKQESQLRNEVAILQNLHHPGVVNLECMFETPERVFVVME
KLHGDMLEMILSSEKGRLPEHITKFLITQILVALRHLHFKNIVHCDLKPENVLLASADPF
PQVKLCDFGFARIIGEKSFRRSVVGTPAYLAPEVLRNKGYNRSLDMWSVGVIIYVSLSGT
FPFNEDEDIHDQIQNAAFMYPPNPWKEISHEAIDLINNLLQVKMRKRYSVDKTLSHPWLQ
DYQTWLDLRELECKIGERYITHESDDLRWEKYAGEQGLQYPTHLINPSASHSDTPETEET
EMKALGERVSIL
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| BDBM32360 |
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| n/a |
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| Name | BDBM32360 |
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| Synonyms: | (3,5-dichloro-2-pyridyl)-[1-(2-pyridyl)ethylideneamino]amine | 3,5-bis(chloranyl)-N-(1-pyridin-2-ylethylideneamino)pyridin-2-amine | 3,5-dichloro-N-(1-pyridin-2-ylethylideneamino)pyridin-2-amine | 3,5-dichloro-N-[1-(2-pyridinyl)ethylideneamino]-2-pyridinamine | MLS000772548 | SMR000377273 | cid_3351416 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H10Cl2N4 |
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| Mol. Mass. | 281.141 |
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| SMILES | CC(N=Nc1ncc(Cl)cc1Cl)c1ccccn1 |w:3.3| |
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| Structure | 
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